Compile Data Set for Download or QSAR
Report error Found 187 Enz. Inhib. hit(s) with all data for entry = 50042444
TargetMuscarinic acetylcholine receptor M3(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50194640((2R)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluoroph...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to human M3 muscarinic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426242(CHEMBL2312346)
Affinity DataIC50: 0.450nMAssay Description:Orthosteric antagonist activity at M5 muscarinic receptor in rat striatal slices assessed as inhibition of 100 uM oxotremorine-evoked [3H]DA releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50111346(SCH-211803 | (2-Amino-3-methyl-phenyl)-{4-[4-(3-ch...)
Affinity DataKi:  0.890nMAssay Description:Binding affinity to human M2 muscarinic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426284(CHEMBL326450)
Affinity DataKi:  1nMAssay Description:Binding affinity to human M4 muscarinic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50368127(Isoptpo Hyoscine | SCOPOLAMINE)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]NMS from human M3 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50368127(Isoptpo Hyoscine | SCOPOLAMINE)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]NMS from human M1 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50073501(CHEMBL120119 | CHEMBL1180285 | 1-Ethyl-4-phenyl-1,...)
Affinity DataIC50: 8.80nMAssay Description:Binding affinity to human M1 muscarinic receptor expressed in cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM39341(PIRENZEPINE DIHYDROCHLORIDE | SMR000058502 | MLS00...)
Affinity DataKi:  9.10nMAssay Description:Binding affinity to human M1 muscarinic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50368127(Isoptpo Hyoscine | SCOPOLAMINE)
Affinity DataKi:  9.5nMAssay Description:Displacement of [3H]NMS from human M2 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50368127(Isoptpo Hyoscine | SCOPOLAMINE)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]NMS from human M5 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426256(CHEMBL2312358)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]NMS from human M1 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50073501(CHEMBL120119 | CHEMBL1180285 | 1-Ethyl-4-phenyl-1,...)
Affinity DataIC50: 25nMAssay Description:Binding affinity to human M5 muscarinic receptor expressed in cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426256(CHEMBL2312358)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]NMS from human M5 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50368127(Isoptpo Hyoscine | SCOPOLAMINE)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]NMS from human M4 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50194640((2R)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluoroph...)
Affinity DataKi:  42nMAssay Description:Binding affinity to human M4 muscarinic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426253(CHEMBL2312361)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]NMS from human M5 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426264(CHEMBL2312378)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]NMS from human M1 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50111346(SCH-211803 | (2-Amino-3-methyl-phenyl)-{4-[4-(3-ch...)
Affinity DataKi:  61nMAssay Description:Binding affinity to human M4 muscarinic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426244(CHEMBL2312370)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]NMS from human M5 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataKi:  81nMAssay Description:Binding affinity to human M2 muscarinic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50111346(SCH-211803 | (2-Amino-3-methyl-phenyl)-{4-[4-(3-ch...)
Affinity DataKi:  85nMAssay Description:Binding affinity to human M5 muscarinic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50073501(CHEMBL120119 | CHEMBL1180285 | 1-Ethyl-4-phenyl-1,...)
Affinity DataIC50: 88nMAssay Description:Binding affinity to human M3 muscarinic receptor expressed in cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426271(CHEMBL2312392)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]NMS from human M1 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM39341(PIRENZEPINE DIHYDROCHLORIDE | SMR000058502 | MLS00...)
Affinity DataKi:  105nMAssay Description:Binding affinity to human M4 muscarinic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426246(CHEMBL2312368)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]NMS from human M5 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426264(CHEMBL2312378)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]NMS from human M5 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM39341(PIRENZEPINE DIHYDROCHLORIDE | SMR000058502 | MLS00...)
Affinity DataKi:  126nMAssay Description:Binding affinity to human M5 muscarinic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50073501(CHEMBL120119 | CHEMBL1180285 | 1-Ethyl-4-phenyl-1,...)
Affinity DataIC50: 136nMAssay Description:Binding affinity to human M2 muscarinic receptor expressed in cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50073501(CHEMBL120119 | CHEMBL1180285 | 1-Ethyl-4-phenyl-1,...)
Affinity DataIC50: 138nMAssay Description:Binding affinity to human M4 muscarinic receptor expressed in cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426258(CHEMBL2312384)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]NMS from human M1 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426259(CHEMBL2312383)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]NMS from human M5 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426276(CHEMBL2312387)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]NMS from human M5 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426284(CHEMBL326450)
Affinity DataKi:  151nMAssay Description:Binding affinity to human M3 muscarinic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM39341(PIRENZEPINE DIHYDROCHLORIDE | SMR000058502 | MLS00...)
Affinity DataKi:  158nMAssay Description:Binding affinity to human M3 muscarinic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50073489(CHEMBL1180343 | CHEMBL123099 | 1-Ethyl-4-phenyl-1,...)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]NMS from human M1 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50194640((2R)-1-((2S,4R)-4-hydroxy-1-[3,3,3-tris(4-fluoroph...)
Affinity DataKi:  170nMAssay Description:Binding affinity to human M1 muscarinic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426271(CHEMBL2312392)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]NMS from human M5 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426258(CHEMBL2312384)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]NMS from human M5 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426247(CHEMBL2312367)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]NMS from human M5 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426272(CHEMBL2312391)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]NMS from human M1 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426265(CHEMBL2312377)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]NMS from human M1 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426280(CHEMBL2312344)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]NMS from human M1 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426266(CHEMBL2312376)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]NMS from human M5 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426269(CHEMBL2312373)
Affinity DataKi:  240nMAssay Description:Displacement of [3H]NMS from human M1 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426265(CHEMBL2312377)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]NMS from human M5 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426245(CHEMBL2312369)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]NMS from human M5 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426253(CHEMBL2312361)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]NMS from human M1 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426272(CHEMBL2312391)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]NMS from human M5 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426244(CHEMBL2312370)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]NMS from human M1 muscarinic receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50426284(CHEMBL326450)
Affinity DataKi:  339nMAssay Description:Binding affinity to human M2 muscarinic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
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