Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50042999
TargetMicrotubule-associated protein tau(Human)
Humboldt Universit£T Zu Berlin

Curated by ChEMBL
LigandPNGBDBM50430742(Toluidine Blue O | Blutene | TOLONIUM CHLORIDE)
Affinity DataIC50: 69nMAssay Description:Inhibition of tau protein aggregation (unknown origin) at 5:1 compound to protein concentration by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Humboldt Universit£T Zu Berlin

Curated by ChEMBL
LigandPNGBDBM50434370(GNF-Pf-3564 | CHEMBL593252 | Thionin (14))
Affinity DataIC50: 69nMAssay Description:Inhibition of tau protein aggregation (unknown origin) at 5:1 compound to protein concentration by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Humboldt Universit£T Zu Berlin

Curated by ChEMBL
LigandPNGBDBM50434371(AZURE A | Azure A (12))
Affinity DataIC50: 69nMAssay Description:Inhibition of tau protein aggregation (unknown origin) at 5:1 compound to protein concentration by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Humboldt Universit£T Zu Berlin

Curated by ChEMBL
LigandPNGBDBM50434366(CHEMBL1789430)
Affinity DataIC50: 80nMAssay Description:Inhibition of tau protein aggregation (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Humboldt Universit£T Zu Berlin

Curated by ChEMBL
LigandPNGBDBM32299(cid_12004742 | MLS000559792 | 3-(2-Hydroxy-ethyl)-...)
Affinity DataIC50: 380nMAssay Description:Inhibition of tau protein aggregation (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Humboldt Universit£T Zu Berlin

Curated by ChEMBL
LigandPNGBDBM50434368(CHEMBL2386876)
Affinity DataIC50: 970nMAssay Description:Inhibition of tau protein aggregation (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Humboldt Universit£T Zu Berlin

Curated by ChEMBL
LigandPNGBDBM15236(CHEMBL164 | Cannabiscetin | 3,5,7-trihydroxy-2-(3,...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant brain tau protein (412 amino acid residues) filament assembly expressed in Escherichia coli BL21(DE3) by electron mic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Humboldt Universit£T Zu Berlin

Curated by ChEMBL
LigandPNGBDBM50070942((-)-Epigallocatechin-3-o-gallate | (-)-Epigallocat...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human recombinant brain tau protein (412 amino acid residues) filament assembly expressed in Escherichia coli BL21(DE3) by electron mic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Humboldt Universit£T Zu Berlin

Curated by ChEMBL
LigandPNGBDBM50434369(Methylthioninium Chloride | Methylene Blue | Methy...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human recombinant brain tau protein (412 amino acid residues) filament assembly expressed in Escherichia coli BL21(DE3) by electron mic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Humboldt Universit£T Zu Berlin

Curated by ChEMBL
LigandPNGBDBM50434371(AZURE A | Azure A (12))
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human recombinant brain tau protein (412 amino acid residues) filament assembly expressed in Escherichia coli BL21(DE3) by electron mic...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMicrotubule-associated protein tau(Human)
Humboldt Universit£T Zu Berlin

Curated by ChEMBL
LigandPNGBDBM50434369(Methylthioninium Chloride | Methylene Blue | Methy...)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of tau protein aggregation (unknown origin) by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed