Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50005386
TargetGastrin/cholecystokinin type B receptor(Human)
Pierre and Marie Curie University

Curated by ChEMBL
LigandPNGBDBM50491639(CHEMBL2386885)
Affinity DataIC50: 5.20nMAssay Description:Displacement of Eu-DTPA-CCK8 from CCK2 receptor in HEK293 cells after 2 hrs by TRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pierre and Marie Curie University

Curated by ChEMBL
LigandPNGBDBM50491638(CHEMBL2386887)
Affinity DataIC50: 6nMAssay Description:Displacement of Eu-DTPA-CCK8 from CCK2 receptor in HEK293 cells after 2 hrs by TRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pierre and Marie Curie University

Curated by ChEMBL
LigandPNGBDBM50491641(CHEMBL2386886)
Affinity DataIC50: 8.5nMAssay Description:Displacement of Eu-DTPA-CCK8 from CCK2 receptor in HEK293 cells after 2 hrs by TRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pierre and Marie Curie University

Curated by ChEMBL
LigandPNGBDBM50491636(CHEMBL2386884)
Affinity DataIC50: 12nMAssay Description:Displacement of Eu-DTPA-CCK8 from CCK2 receptor in HEK293 cells after 2 hrs by TRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Pierre and Marie Curie University

Curated by ChEMBL
LigandPNGBDBM50491635(CHEMBL2386882)
Affinity DataIC50: 12nMAssay Description:Binding affinity to MC4R in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pierre and Marie Curie University

Curated by ChEMBL
LigandPNGBDBM50491637(CHEMBL2386888)
Affinity DataIC50: 16nMAssay Description:Displacement of Eu-DTPA-CCK8 from CCK2 receptor in HEK293 cells after 2 hrs by TRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Pierre and Marie Curie University

Curated by ChEMBL
LigandPNGBDBM50491640(CHEMBL2386883)
Affinity DataIC50: 40nMAssay Description:Binding affinity to MC4R in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pierre and Marie Curie University

Curated by ChEMBL
LigandPNGBDBM50491640(CHEMBL2386883)
Affinity DataIC50: 4.60E+6nMAssay Description:Displacement of Eu-DTPA-CCK8 from CCK2 receptor in HEK293 cells after 2 hrs by TRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed