Report error Found 277 Enz. Inhib. hit(s) with all data for entry = 50043068
TargetDual specificity protein kinase CLK1(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of CLK4 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of DYRK1B (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of CLK4 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of DYRK1B (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of CLK4 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of CLK4 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Mouse)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of mouse recombinant GST-tagged CLK4 expressed in Escherichia coli DH5[alpha] using NH2-RSPSYGRSRSRSRSRSRSRSRSNSRSRSY-OH as substrate by l...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of CLK4 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of DYRK1B (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of DYRK1B (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of CLK4 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of CLK4 (unknown origin) by bioluminescence assayMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of CLK2 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of human recombinant CLK1 (148 to 484 amino acids) expressed in Escherichia coli BL21(DE3) using AFRREWSPGKEAKK as substrate preincubated ...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mouse)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of mouse recombinant GST-tagged CLK1 expressed in Escherichia coli DH5[alpha] using NH2-RSPSYGRSRSRSRSRSRSRSRSNSRSRSY-OH as substrate by l...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of CLK2 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of CLK4 (unknown origin) by bioluminescence assayMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of CLK4 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of CLK4 (unknown origin) by bioluminescence assayMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of CLK2 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of DYRK1B (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibition of CLK2 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of CLK4 (unknown origin) by bioluminescence assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of DYRK1A (unknown origin) by bioluminescence assayMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of CLK4 (unknown origin) by bioluminescence assayMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of CLK4 (unknown origin) by bioluminescence assayMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of CLK2 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of DYRK1B (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of CLK4 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of DYRK1A (unknown origin) by bioluminescence assayMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of CLK4 (unknown origin) by bioluminescence assayMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of CLK4 (unknown origin) by bioluminescence assayMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of CLK2 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of DYRK1B (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
University of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of DYRK1A (unknown origin) using YRASPSRPESPRPPA-NH2 as substrate preincubated for 10 mins prior to substrate addition by LDH assayMore data for this Ligand-Target Pair
