Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50005481
TargetKelch-like ECH-associated protein 1(Human)
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50492323(CHEMBL2402205)
Affinity DataIC50: 33nMAssay Description:Displacement of MR121-Nrf2 from human N-terminal His-tagged Kelch-DC domain of Keap1 (321 to 609) expressed in Escherichia coli BL21 (DE3) after 40 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50006931(CHEMBL2402207)
Affinity DataIC50: 2.70E+3nMAssay Description:Displacement of MR121-Nrf2 from human N-terminal His-tagged Kelch-DC domain of Keap1 (321 to 609) expressed in Escherichia coli BL21 (DE3) after 40 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetKelch-like ECH-associated protein 1(Human)
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50120421(CHEMBL2402206)
Affinity DataIC50: 1.18E+5nMAssay Description:Displacement of MR121-Nrf2 from human N-terminal His-tagged Kelch-DC domain of Keap1 (321 to 609) expressed in Escherichia coli BL21 (DE3) after 40 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)