Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50043114
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436176(Dynacirc | Dynacirc Cr | Isrodipine | PN-200-110 |...)
Affinity DataIC50: 107nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436175(CHEMBL2381007)
Affinity DataIC50: 170nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436171(CHEMBL2398404)
Affinity DataIC50: 350nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436174(CHEMBL2398408)
Affinity DataIC50: 410nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436173(CHEMBL2398396)
Affinity DataIC50: 420nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436172(CHEMBL2398418)
Affinity DataIC50: 500nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436171(CHEMBL2398404)
Affinity DataIC50: 500nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436170(CHEMBL2398425)
Affinity DataIC50: 580nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436167(CHEMBL2398406)
Affinity DataIC50: 640nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436169(CHEMBL2398409)
Affinity DataIC50: 860nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436168(CHEMBL2398401)
Affinity DataIC50: 1.02E+3nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436167(CHEMBL2398406)
Affinity DataIC50: 1.02E+3nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436199(CHEMBL2398399)
Affinity DataIC50: 1.81E+3nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436198(CHEMBL2398422)
Affinity DataIC50: 1.93E+3nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436197(CHEMBL2398402)
Affinity DataIC50: 2.36E+3nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436196(CHEMBL2398400)
Affinity DataIC50: 2.45E+3nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436181(CHEMBL2398403)
Affinity DataIC50: 2.48E+3nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436195(CHEMBL2398419)
Affinity DataIC50: 2.48E+3nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436194(CHEMBL2398407)
Affinity DataIC50: 3.07E+3nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50035789(6-Methyl-2-methylsulfanyl-4-(3-nitro-phenyl)-1,4-d...)
Affinity DataIC50: 3.29E+3nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436193(CHEMBL2398393)
Affinity DataIC50: 4.23E+3nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436192(CHEMBL2398394)
Affinity DataIC50: 4.75E+3nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436191(CHEMBL2398398)
Affinity DataIC50: 5.54E+3nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436190(CHEMBL2398395)
Affinity DataIC50: 6.11E+3nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436189(CHEMBL2398423)
Affinity DataIC50: 6.13E+3nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436188(CHEMBL2398405)
Affinity DataIC50: 9.87E+3nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436187(CHEMBL2398420)
Affinity DataIC50: 1.04E+4nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436186(CHEMBL2398413)
Affinity DataIC50: 1.07E+4nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436185(CHEMBL2398410)
Affinity DataIC50: 1.17E+4nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436184(CHEMBL2398424)
Affinity DataIC50: 1.39E+4nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436183(CHEMBL2398416)
Affinity DataIC50: 1.48E+4nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436182(CHEMBL2398397)
Affinity DataIC50: 1.61E+4nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436181(CHEMBL2398403)
Affinity DataIC50: 2.17E+4nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436180(CHEMBL2398412)
Affinity DataIC50: 5.50E+4nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436179(CHEMBL2398417)
Affinity DataIC50: 5.66E+4nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436178(CHEMBL167975)
Affinity DataIC50: 5.81E+4nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Rabbit)
Northwestern University

Curated by ChEMBL
LigandPNGBDBM50436177(CHEMBL2398411)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at rabbit voltage-dependent L-type calcium channel Cav1.2alpha-1C expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed