Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50043154
TargetHistamine H1 receptor(Human)
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292603(2-(pyrrolidin-1-yl)ethyl 10H-phenothiazine-10-carb...)
Affinity DataKi:  29nMAssay Description:Antagonist activity at histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292604(3-(diethylamino)propyl 10H-phenothiazine-10-carbox...)
Affinity DataKi:  430nMAssay Description:Antagonist activity at histamine H1 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistamine H2 receptor(Human)
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292603(2-(pyrrolidin-1-yl)ethyl 10H-phenothiazine-10-carb...)
Affinity DataKi:  540nMAssay Description:Antagonist activity at histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistamine H2 receptor(Human)
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292604(3-(diethylamino)propyl 10H-phenothiazine-10-carbox...)
Affinity DataKi:  1.40E+3nMAssay Description:Antagonist activity at histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292603(2-(pyrrolidin-1-yl)ethyl 10H-phenothiazine-10-carb...)
Affinity DataKi:  1.90E+3nMAssay Description:Antagonist activity at serotonin 5HT3 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50292604(3-(diethylamino)propyl 10H-phenothiazine-10-carbox...)
Affinity DataKi:  3.90E+3nMAssay Description:Antagonist activity at serotonin 5HT3 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistamine H2 receptor(Human)
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50219223(1-(10H-phenothiazin-10-yl)-4-phenylbutan-1-one | C...)
Affinity DataKi:  7.50E+3nMAssay Description:Antagonist activity at histamine H2 receptor (unknown origin) by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed