Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50001495
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015924(CHEMBL83564 | 3-Acetoxymethyl-7-methoxy-5,5,8-trio...)
Affinity DataIC50: 40nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015916(CHEMBL83565 | 3-Acetoxymethyl-7-methoxy-5,5,8-trio...)
Affinity DataIC50: 70nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015900(CHEMBL315714 | 3-Acetoxymethyl-7-methoxy-5,5,8-tri...)
Affinity DataIC50: 100nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015922(CHEMBL315377 | 3-Acetoxymethyl-7-methoxy-5,5,8-tri...)
Affinity DataIC50: 100nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015913(CHEMBL314155 | Acetic acid 2-(benzyl-methyl-carbam...)
Affinity DataIC50: 100nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015912(CHEMBL315690 | 3-Acetoxymethyl-7-methoxy-5,5,8-tri...)
Affinity DataIC50: 100nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015904(CHEMBL312327 | 3-Acetoxymethyl-7-methoxy-5,5,8-tri...)
Affinity DataIC50: 100nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015907(CHEMBL432765 | [(3-Acetoxymethyl-7-methoxy-5,5,8-t...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015921(CHEMBL315829 | 3-Acetoxymethyl-7-methoxy-5,5,8-tri...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015920(CHEMBL85215 | 3-Acetoxymethyl-7-methoxy-5,5,8-trio...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015909(CHEMBL86173 | 3-Acetoxymethyl-7-methoxy-5,5,8-trio...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015919(CHEMBL314845 | 4-[(3-Acetoxymethyl-7-methoxy-5,5,8...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015914(CHEMBL440309 | (6R,7S)-3-Acetoxymethyl-7-methoxy-5...)
Affinity DataIC50: 400nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015923(CHEMBL314821 | 3-Acetoxymethyl-7-methoxy-5,5,8-tri...)
Affinity DataIC50: 400nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015901(CHEMBL85563 | 3-Acetoxymethyl-7-methoxy-5,5,8-trio...)
Affinity DataIC50: 400nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015915(4-{[((6R,7S)-3-Acetoxymethyl-7-methoxy-5,5,8-triox...)
Affinity DataIC50: 400nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015918(CHEMBL313667 | 3-Acetoxymethyl-7-methoxy-5,5,8-tri...)
Affinity DataIC50: 500nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015917(CHEMBL84839 | 3-Acetoxymethyl-7-methoxy-5,5,8-trio...)
Affinity DataIC50: 800nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015910(CHEMBL86142 | Acetic acid 2-tert-butylcarbamoyl-7-...)
Affinity DataIC50: 800nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015879(CHEMBL84724 | 3-Acetoxymethyl-7-methoxy-5,5,8-trio...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015902(CHEMBL312174 | 3-[(3-Acetoxymethyl-7-methoxy-5,5,8...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015905(CHEMBL86037 | Acetic acid 2-dimethylcarbamoyl-7-me...)
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015903(CHEMBL306251 | [(3-Acetoxymethyl-7-methoxy-5,5,8-t...)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015906(CHEMBL313991 | Acetic acid 2-benzylcarbamoyl-7-met...)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015911(CHEMBL310583 | 3-[(3-Acetoxymethyl-7-methoxy-5,5,8...)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015908(CHEMBL312438 | [(3-Acetoxymethyl-7-methoxy-5,5,8-t...)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Merck Sharp and Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50015899(CHEMBL314721 | 3-Acetoxymethyl-7-methoxy-5,5,8-tri...)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro inhibition of Human Leukocyte Elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed