Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50043476
TargetTGF-beta receptor type-1(Human)
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50441661(CHEMBL2435034)
Affinity DataIC50: 240nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50110208(SB-431542 | cid_4521392 | 4-(5-(benzo[d][1,3]dioxo...)
Affinity DataIC50: 350nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50441660(CHEMBL2435035)
Affinity DataIC50: 650nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50441659(CHEMBL2435036)
Affinity DataIC50: 800nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50441662(CHEMBL2435041)
Affinity DataIC50: 950nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50441666(CHEMBL2435044)
Affinity DataIC50: 990nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50441663(CHEMBL2435040)
Affinity DataIC50: 1.78E+3nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50441664(CHEMBL2435039)
Affinity DataIC50: 2.08E+3nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50441667(CHEMBL2435043)
Affinity DataIC50: 2.43E+3nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50441665(CHEMBL2435045)
Affinity DataIC50: 3.36E+3nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTGF-beta receptor type-1(Human)
Capital Normal University

Curated by ChEMBL
LigandPNGBDBM50441658(CHEMBL2435037)
Affinity DataIC50: 3.82E+3nMAssay Description:Inhibition of TGFbeta-induced downstream transcriptional activation of ALK5 (unknown origin) expressed in CHO-HIR cells assessed as intracellular tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed