Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 6014
TargetDeath-associated protein kinase 1(Human)
Duke University Medical Center

LigandPNGBDBM104065(HS38)
Affinity DataKd:  79nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Duke University Medical Center

LigandPNGBDBM104065(HS38)
Affinity DataIC50: 200nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetDeath-associated protein kinase 1(Human)
Duke University Medical Center

LigandPNGBDBM104065(HS38)
Affinity DataIC50: 200nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetDeath-associated protein kinase 1(Human)
Duke University Medical Center

LigandPNGBDBM104065(HS38)
Affinity DataKd:  280nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetDeath-associated protein kinase 1(Human)
Duke University Medical Center

LigandPNGBDBM104065(HS38)
Affinity DataKd:  300nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetDeath-associated protein kinase 1(Human)
Duke University Medical Center

LigandPNGBDBM104066(HS43)
Affinity DataKd:  320nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Duke University Medical Center

LigandPNGBDBM104065(HS38)
Affinity DataKd:  810nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Duke University Medical Center

LigandPNGBDBM104065(HS38)
Affinity DataIC50: 1.40E+3nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetDeath-associated protein kinase 1(Human)
Duke University Medical Center

LigandPNGBDBM104066(HS43)
Affinity DataKd:  1.50E+3nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetDeath-associated protein kinase 1(Human)
Duke University Medical Center

LigandPNGBDBM104066(HS43)
Affinity DataKd:  1.50E+3nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Duke University Medical Center

LigandPNGBDBM104066(HS43)
Affinity DataKd:  1.60E+3nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Duke University Medical Center

LigandPNGBDBM104065(HS38)
Affinity DataIC50: 1.70E+3nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
LigandPNGBDBM104065(HS38)
Affinity DataIC50: 1.80E+3nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Duke University Medical Center

LigandPNGBDBM104065(HS38)
Affinity DataKd:  1.80E+3nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Duke University Medical Center

LigandPNGBDBM104066(HS43)
Affinity DataKd:  1.80E+3nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Duke University Medical Center

LigandPNGBDBM104066(HS43)
Affinity DataKd:  3.20E+3nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Duke University Medical Center

LigandPNGBDBM104065(HS38)
Affinity DataKd:  6.50E+3nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
Duke University Medical Center

LigandPNGBDBM104065(HS38)
Affinity DataIC50: 1.80E+4nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetMyosin light chain kinase, smooth muscle(Human)
Duke University Medical Center

LigandPNGBDBM104065(HS38)
Affinity DataIC50: 1.90E+4nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Duke University Medical Center

LigandPNGBDBM104065(HS38)
Affinity DataIC50: 2.00E+5nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed