Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50005728
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50444438(CHEMBL2442495)
Affinity DataIC50: 50nMAssay Description:Antagonist activity at human EP1 receptor by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493974(CHEMBL2442494)
Affinity DataIC50: 84nMAssay Description:Antagonist activity at human EP1 receptor by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493969(CHEMBL2442490)
Affinity DataIC50: 180nMAssay Description:Antagonist activity at human EP1 receptor by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50444438(CHEMBL2442495)
Affinity DataKi:  290nMAssay Description:Binding affinity to human EP1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50250685(CHEMBL1479261 | US10961200, Compound 62 | US112479...)
Affinity DataIC50: 320nMAssay Description:Antagonist activity at human EP1 receptor by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493970(CHEMBL2442488)
Affinity DataIC50: 320nMAssay Description:Antagonist activity at human EP1 receptor by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493971(CHEMBL2442486)
Affinity DataIC50: 430nMAssay Description:Antagonist activity at human EP1 receptor by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493972(CHEMBL2442497)
Affinity DataIC50: 500nMAssay Description:Antagonist activity at human EP1 receptor by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50444438(CHEMBL2442495)
Affinity DataIC50: 500nMAssay Description:Antagonist activity at human EP1 receptor by intracellular Ca2+ release assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493969(CHEMBL2442490)
Affinity DataKi:  530nMAssay Description:Binding affinity to human EP1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493973(CHEMBL2442489)
Affinity DataIC50: 580nMAssay Description:Antagonist activity at human EP1 receptor by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493969(CHEMBL2442490)
Affinity DataIC50: 800nMAssay Description:Antagonist activity at human EP1 receptor by intracellular Ca2+ release assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493968(CHEMBL2442485)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human EP1 receptor by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493968(CHEMBL2442485)
Affinity DataKi: >2.70E+3nMAssay Description:Binding affinity to human EP4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493969(CHEMBL2442490)
Affinity DataKi: >2.70E+3nMAssay Description:Binding affinity to human EP4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493968(CHEMBL2442485)
Affinity DataIC50: 2.70E+3nMAssay Description:Antagonist activity at EP4 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50444438(CHEMBL2442495)
Affinity DataKi: >2.70E+3nMAssay Description:Binding affinity to human EP4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493975(CHEMBL2442487)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at human EP1 receptor by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493968(CHEMBL2442485)
Affinity DataIC50: 5.00E+3nMAssay Description:Antagonist activity at EP3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493968(CHEMBL2442485)
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity to human EP3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493969(CHEMBL2442490)
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity to human EP3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50444438(CHEMBL2442495)
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity to human EP3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493968(CHEMBL2442485)
Affinity DataIC50: 5.80E+3nMAssay Description:Antagonist activity at human EP1 receptor by intracellular Ca2+ release assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493968(CHEMBL2442485)
Affinity DataKi: >8.00E+3nMAssay Description:Binding affinity to human EP2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493968(CHEMBL2442485)
Affinity DataIC50: 8.00E+3nMAssay Description:Antagonist activity at EP2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493969(CHEMBL2442490)
Affinity DataKi: >8.00E+3nMAssay Description:Binding affinity to human EP2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50444438(CHEMBL2442495)
Affinity DataKi: >8.00E+3nMAssay Description:Binding affinity to human EP2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50493968(CHEMBL2442485)
Affinity DataKi:  8.70E+3nMAssay Description:Binding affinity to human EP1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed