Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50005837
TargetSodium-dependent serotonin transporter(Rat)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM25870(CITALOPRAM HYDROBROMIDE | [3H]Escitalopram | Escit...)
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]paroxetine from SERT in rat cortical membranes after 6 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataIC50: 6nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50494871(CHEMBL3092348)
Affinity DataIC50: 13nMAssay Description:Displacement of [3H]paroxetine from SERT in rat cortical membranes after 6 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50494864(CHEMBL3092343)
Affinity DataIC50: 14nMAssay Description:Displacement of [3H]paroxetine from SERT in rat cortical membranes after 6 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50494870(CHEMBL3092351)
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50494869(CHEMBL3092342)
Affinity DataIC50: 16nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50494869(CHEMBL3092342)
Affinity DataIC50: 26nMAssay Description:Displacement of [3H]paroxetine from SERT in rat cortical membranes after 6 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50494873(CHEMBL3092347)
Affinity DataIC50: 37nMAssay Description:Displacement of [3H]paroxetine from SERT in rat cortical membranes after 6 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50494865(CHEMBL3092346)
Affinity DataIC50: 39nMAssay Description:Displacement of [3H]paroxetine from SERT in rat cortical membranes after 6 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50494868(CHEMBL3092344)
Affinity DataIC50: 43nMAssay Description:Displacement of [3H]paroxetine from SERT in rat cortical membranes after 6 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50494867(CHEMBL3092345)
Affinity DataIC50: 61nMAssay Description:Displacement of [3H]paroxetine from SERT in rat cortical membranes after 6 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50494872(CHEMBL3092350)
Affinity DataIC50: 87nMAssay Description:Displacement of [3H]paroxetine from SERT in rat cortical membranes after 6 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50494866(CHEMBL3092349)
Affinity DataIC50: 98nMAssay Description:Displacement of [3H]paroxetine from SERT in rat cortical membranes after 6 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50494865(CHEMBL3092346)
Affinity DataIC50: 128nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50494870(CHEMBL3092351)
Affinity DataIC50: 137nMAssay Description:Displacement of [3H]paroxetine from SERT in rat cortical membranes after 6 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50494866(CHEMBL3092349)
Affinity DataIC50: 599nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50494872(CHEMBL3092350)
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50494873(CHEMBL3092347)
Affinity DataIC50: 2.70E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50494868(CHEMBL3092344)
Affinity DataIC50: 4.50E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50494867(CHEMBL3092345)
Affinity DataIC50: 4.90E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50494871(CHEMBL3092348)
Affinity DataIC50: 5.70E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universidad De Chile

Curated by ChEMBL
LigandPNGBDBM50494864(CHEMBL3092343)
Affinity DataIC50: 7.20E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed