Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50043699
TargetBeta-2 adrenergic receptor(Guinea pig)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50444835(CHEMBL3099249)
Affinity DataEC50:  1nMAssay Description:Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50444836(CHEMBL3099248)
Affinity DataEC50:  5nMAssay Description:Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50444837(CHEMBL3099251)
Affinity DataEC50:  13nMAssay Description:Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50444838(CHEMBL3099250)
Affinity DataEC50:  10nMAssay Description:Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50151720(CHEMBL605993 | Symbicort | cid_9912089 | N-(2-hydr...)
Affinity DataEC50:  0.126nMAssay Description:Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBeta-2 adrenergic receptor(Guinea pig)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  32nMAssay Description:Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50444835(CHEMBL3099249)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50444836(CHEMBL3099248)
Affinity DataEC50:  5nMAssay Description:Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50444837(CHEMBL3099251)
Affinity DataEC50:  13nMAssay Description:Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50444838(CHEMBL3099250)
Affinity DataEC50:  10nMAssay Description:Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50151720(CHEMBL605993 | Symbicort | cid_9912089 | N-(2-hydr...)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBeta-2 adrenergic receptor(Guinea pig)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  32nMAssay Description:Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed