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Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50005914
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495365(CHEMBL3110241)
Affinity DataKd:  8.00E+3nMAssay Description:Binding affinity to human BAZ2B expressed in Escherichia coli BL21(DE3) by direct isothermal titration calorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495365(CHEMBL3110241)
Affinity DataIC50: 9.00E+3nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495361(CHEMBL3110228)
Affinity DataKd:  1.00E+4nMAssay Description:Binding affinity to human BAZ2B expressed in Escherichia coli BL21(DE3) by competitive isothermal titration calorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495361(CHEMBL3110228)
Affinity DataIC50: 1.20E+4nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495368(CHEMBL3110242)
Affinity DataIC50: 1.40E+4nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495368(CHEMBL3110242)
Affinity DataKd:  1.70E+4nMAssay Description:Binding affinity to human BAZ2B expressed in Escherichia coli BL21(DE3) by direct isothermal titration calorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495371(CHEMBL3110247)
Affinity DataIC50: 2.40E+4nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495390(CHEMBL3110249)
Affinity DataIC50: 2.50E+4nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495385(CHEMBL1542917)
Affinity DataIC50: 2.60E+4nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495373(CHEMBL3110262)
Affinity DataIC50: 3.60E+4nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495372(CHEMBL1526788)
Affinity DataIC50: 3.70E+4nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495384(CHEMBL3110229)
Affinity DataIC50: 3.70E+4nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495371(CHEMBL3110247)
Affinity DataIC50: 3.70E+4nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50207717(CHEMBL3110243)
Affinity DataIC50: 3.80E+4nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495386(CHEMBL3110256)
Affinity DataIC50: 4.60E+4nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495364(CHEMBL3110257)
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495375(CHEMBL3110258)
Affinity DataIC50: 5.50E+4nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495371(CHEMBL3110247)
Affinity DataKd:  6.50E+4nMAssay Description:Binding affinity to human BAZ2B expressed in Escherichia coli BL21(DE3) by competitive isothermal titration calorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495387(CHEMBL3110250)
Affinity DataIC50: 6.60E+4nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495376(CHEMBL3110253)
Affinity DataIC50: 6.90E+4nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495363(CHEMBL3110239)
Affinity DataKd: >1.00E+5nMAssay Description:Binding affinity to human BAZ2B expressed in Escherichia coli BL21(DE3) by direct isothermal titration calorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495374(CHEMBL3110261)
Affinity DataIC50: 1.02E+5nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495381(CHEMBL3110244)
Affinity DataIC50: 1.09E+5nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495377(CHEMBL3110251)
Affinity DataIC50: 1.43E+5nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495382(CHEMBL3110252)
Affinity DataIC50: 1.52E+5nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495380(CHEMBL2441350)
Affinity DataIC50: 1.90E+5nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495389(CHEMBL3110245)
Affinity DataIC50: 2.41E+5nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495383(CHEMBL3110255)
Affinity DataKd:  2.74E+5nMAssay Description:Binding affinity to human BAZ2B expressed in Escherichia coli BL21(DE3) by competitive isothermal titration calorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495388(CHEMBL1650611)
Affinity DataIC50: 2.79E+5nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495370(CHEMBL3110254)
Affinity DataKd:  3.36E+5nMAssay Description:Binding affinity to human BAZ2B expressed in Escherichia coli BL21(DE3) by competitive isothermal titration calorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495379(CHEMBL1568712)
Affinity DataIC50: 4.76E+5nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495378(CHEMBL3110248)
Affinity DataIC50: 4.95E+5nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495380(CHEMBL2441350)
Affinity DataKd:  5.24E+5nMAssay Description:Binding affinity to human BAZ2B expressed in Escherichia coli BL21(DE3) by direct isothermal titration calorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495369(CHEMBL3110260)
Affinity DataKd:  6.94E+5nMAssay Description:Binding affinity to human BAZ2B expressed in Escherichia coli BL21(DE3) by competitive isothermal titration calorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM181114(US9138393, 4'-(Imidazol-1 yl) acetophenome | US914...)
Affinity DataIC50: 8.26E+5nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495366(CHEMBL3110259)
Affinity DataIC50: 1.00E+6nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495367(CHEMBL3110246)
Affinity DataIC50: 1.09E+6nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495362(CHEMBL3110240)
Affinity DataIC50: 2.00E+6nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed