Compile Data Set for Download or QSAR
Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50005920
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126727(Isoquinoline-5-sulfonic acid 4-{(S)-3-[4-(4-fluoro...)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50404086(CHEMBL341226)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126713(Isoquinoline-5-sulfonic acid 4-{(S)-2-[(isoquinoli...)
Affinity DataIC50: 5.80nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126702(Isoquinoline-5-sulfonic acid 4-{(S)-3-[4-(4-fluoro...)
Affinity DataIC50: 5.80nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50404085(CHEMBL336619)
Affinity DataIC50: 7.90nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50411888(CHEMBL270421)
Affinity DataIC50: 9.10nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415889(CHEMBL1098723)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50404090(CHEMBL424451)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126723(Isoquinoline-5-sulfonic acid 4-{(S)-3-[4-(3-chloro...)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126715(Isoquinoline-5-sulfonic acid 4-[(S)-2-[(isoquinoli...)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126718((S)-4-(3-(4-(2-chlorophenyl)piperazin-1-yl)-2-(N-m...)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50423270(CHEMBL393241)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415882(CHEMBL1094106)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415908(CHEMBL1094641)
Affinity DataIC50: 25nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50423276(CHEMBL396587)
Affinity DataIC50: 27nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126712(Isoquinoline-5-sulfonic acid 4-{(S)-3-[4-(3,4-dich...)
Affinity DataIC50: 34nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50410952(CHEMBL208560)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50423280(CHEMBL245561)
Affinity DataIC50: 49nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415888(CHEMBL1096314)
Affinity DataIC50: 50nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50423272(CHEMBL246578)
Affinity DataIC50: 50nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50495434(CHEMBL131241)
Affinity DataIC50: 63nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415891(CHEMBL1094744)
Affinity DataIC50: 63nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126719(Isoquinoline-5-sulfonic acid 4-{(S)-3-(4-benzyl-pi...)
Affinity DataIC50: 65nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126724(Isoquinoline-5-sulfonic acid 4-{(S)-3-[4-(4-acetyl...)
Affinity DataIC50: 71nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50411878(CHEMBL245754)
Affinity DataIC50: 78nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415909(CHEMBL1094482)
Affinity DataIC50: 79nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50087267((S)-4-(2-(N-methylisoquinoline-5-sulfonamido)-3-ox...)
Affinity DataIC50: 94nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126717(Isoquinoline-5-sulfonic acid 4-{(S)-3-[4-(4-cyano-...)
Affinity DataIC50: 98nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126710(Isoquinoline-5-sulfonic acid 4-{(S)-3-[4-(4-amino-...)
Affinity DataIC50: 101nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126706((S)-4-(3-(4-(4-chlorophenyl)piperazin-1-yl)-2-(N-m...)
Affinity DataIC50: 105nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50404074(CHEMBL337873)
Affinity DataIC50: 126nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415906(CHEMBL1096096)
Affinity DataIC50: 126nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126711(Isoquinoline-5-sulfonic acid 4-{(S)-2-[(isoquinoli...)
Affinity DataIC50: 132nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415898(CHEMBL1096100)
Affinity DataIC50: 158nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415884(CHEMBL1096049)
Affinity DataIC50: 158nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126709(Isoquinoline-5-sulfonic acid 4-{(S)-3-[4-(4-iodo-p...)
Affinity DataIC50: 176nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50423269(CHEMBL245755)
Affinity DataIC50: 191nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415913(CHEMBL1096048)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50423282(CHEMBL246770)
Affinity DataIC50: 209nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50423277(CHEMBL245578)
Affinity DataIC50: 214nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50495436(CHEMBL3108814)
Affinity DataIC50: 251nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415885(CHEMBL1096660)
Affinity DataIC50: 316nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50495438(CHEMBL3108810)
Affinity DataIC50: 398nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50404076(CHEMBL337419)
Affinity DataIC50: 398nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50495437(CHEMBL3108813)
Affinity DataIC50: 501nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415903(CHEMBL1094485)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415900(CHEMBL1095783)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415896(CHEMBL1096030)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415899(CHEMBL1096099)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415893(CHEMBL1095395)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
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