Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50043706
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant AKT1 (unknown origin) using serine/threonine 06 peptide as substrate after 1 hr by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM29511(Pyranonaphthoquinone (PNQ) lactone, 11a)
Affinity DataIC50: 44nMAssay Description:Inhibition of recombinant AKT1 (unknown origin) using serine/threonine 06 peptide as substrate after 1 hr by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50403054(CHEMBL2216825)
Affinity DataIC50: 149nMAssay Description:Inhibition of AKT1 (unknown origin) by high-throughput screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM29517(Pyranonaphthoquinone (PNQ) lactone, 11g)
Affinity DataIC50: 150nMAssay Description:Inhibition of AKT1 (unknown origin) by high-throughput screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM29508(Frenolicin B)
Affinity DataIC50: 198nMAssay Description:Inhibition of AKT1 (unknown origin) by high-throughput screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM29517(Pyranonaphthoquinone (PNQ) lactone, 11g)
Affinity DataIC50: 280nMAssay Description:Inhibition of recombinant AKT1 (unknown origin) using serine/threonine 06 peptide as substrate after 1 hr by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50444880(CHEMBL3099612)
Affinity DataIC50: 2.94E+3nMAssay Description:Inhibition of recombinant AKT1 (unknown origin) using serine/threonine 06 peptide as substrate after 1 hr by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM24776(1,4-dihydronaphthalene-1,4-dione | 1,4-Naphthoquin...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of recombinant AKT1 (unknown origin) using serine/threonine 06 peptide as substrate after 1 hr by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50444877(CHEMBL3099615)
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of recombinant AKT1 (unknown origin) using serine/threonine 06 peptide as substrate after 1 hr by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50444878(CHEMBL3099614)
Affinity DataIC50: 1.37E+4nMAssay Description:Inhibition of recombinant AKT1 (unknown origin) using serine/threonine 06 peptide as substrate after 1 hr by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50444879(CHEMBL3099613)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant AKT1 (unknown origin) using serine/threonine 06 peptide as substrate after 1 hr by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed