Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50006056
TargetSphingosine kinase 1(Human)
The City University of New York

Curated by ChEMBL
LigandPNGBDBM50041978(CHEMBL3134157)
Affinity DataIC50: 28nMAssay Description:Inhibition of recombinant SK1 (unknown origin) using sphingosine and [gamma-32P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSphingosine kinase 1(Human)
The City University of New York

Curated by ChEMBL
LigandPNGBDBM50496601(CHEBI:67106 | (2S,3R)-Sphingosine | CHEMBL1835439)
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of recombinant SK1 (unknown origin) using sphingosine and [gamma-32P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetSphingosine kinase 2(Human)
The City University of New York

Curated by ChEMBL
LigandPNGBDBM50496602(CHEMBL3134155)
Affinity DataIC50: 2.18E+4nMAssay Description:Inhibition of purified SK2 (unknown origin) using sphingosine and [gamma-32P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetSphingosine kinase 1(Human)
The City University of New York

Curated by ChEMBL
LigandPNGBDBM50496603(CHEMBL3134156)
Affinity DataIC50: 2.78E+4nMAssay Description:Inhibition of recombinant SK1 (unknown origin) using sphingosine and [gamma-32P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetSphingosine kinase 1(Human)
The City University of New York

Curated by ChEMBL
LigandPNGBDBM50496602(CHEMBL3134155)
Affinity DataIC50: 6.90E+4nMAssay Description:Inhibition of recombinant SK1 (unknown origin) using sphingosine and [gamma-32P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetSphingosine kinase 2(Human)
The City University of New York

Curated by ChEMBL
LigandPNGBDBM50496603(CHEMBL3134156)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of purified SK2 (unknown origin) using sphingosine and [gamma-32P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetSphingosine kinase 2(Human)
The City University of New York

Curated by ChEMBL
LigandPNGBDBM50496601(CHEBI:67106 | (2S,3R)-Sphingosine | CHEMBL1835439)
Affinity DataIC50: 7.66E+5nMAssay Description:Inhibition of purified SK2 (unknown origin) using sphingosine and [gamma-32P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetSphingosine kinase 2(Human)
The City University of New York

Curated by ChEMBL
LigandPNGBDBM50393642(CHEMBL2158685)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of SK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetSphingosine kinase 2(Human)
The City University of New York

Curated by ChEMBL
LigandPNGBDBM50393641(CHEMBL2158686)
Affinity DataKi:  1.65E+4nMAssay Description:Inhibition of SK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed