Compile Data Set for Download or QSAR
Report error Found 86 Enz. Inhib. hit(s) with all data for entry = 50006024
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496270(CHEMBL3127679)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human histamine H3 receptor expressed in CHOK1 cells after 1.5 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496289(CHEMBL3124968)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human histamine H3 receptor expressed in CHOK1 cells after 1.5 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496294(CHEMBL3127674)
Affinity DataIC50: 0.800nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496273(CHEMBL3127700)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human histamine H3 receptor expressed in CHOK1 cells after 1.5 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496272(CHEMBL3127701)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human histamine H3 receptor expressed in CHOK1 cells after 1.5 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496293(CHEMBL3127676)
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496270(CHEMBL3127679)
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496299(CHEMBL3127675)
Affinity DataIC50: 1.90nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496284(CHEMBL3127691)
Affinity DataIC50: 2.70nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496281(CHEMBL3127698)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human histamine H3 receptor expressed in CHOK1 cells after 1.5 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496296(CHEMBL3127704)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human histamine H3 receptor expressed in CHOK1 cells after 1.5 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496264(CHEMBL3127692)
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496281(CHEMBL3127698)
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496273(CHEMBL3127700)
Affinity DataIC50: 3.60nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496265(CHEMBL3127690)
Affinity DataIC50: 3.60nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496285(CHEMBL3127688)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496260(CHEMBL3127681)
Affinity DataIC50: 4.40nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496271(CHEMBL3127677)
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496266(CHEMBL3127689)
Affinity DataIC50: 6.5nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496289(CHEMBL3124968)
Affinity DataIC50: 8.30nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496290(CHEMBL3127705)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human histamine H3 receptor expressed in CHOK1 cells after 1.5 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496272(CHEMBL3127701)
Affinity DataIC50: 8.80nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496295(CHEMBL3127708)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496297(CHEMBL3127699)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human histamine H3 receptor expressed in CHOK1 cells after 1.5 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496286(CHEMBL3127684)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496280(CHEMBL3127702)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496288(CHEMBL3127687)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496300(CHEMBL3127693)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496292(CHEMBL3127678)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496259(CHEMBL3127672)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human histamine H3 receptor expressed in CHOK1 cells after 1.5 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496276(CHEMBL3127670)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496296(CHEMBL3127704)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496282(CHEMBL3127696)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496263(CHEMBL3127709)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496295(CHEMBL3127708)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human histamine H3 receptor expressed in CHOK1 cells after 1.5 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496297(CHEMBL3127699)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496283(CHEMBL3127694)
Affinity DataIC50: 21nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496276(CHEMBL3127670)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human histamine H3 receptor expressed in CHOK1 cells after 1.5 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496280(CHEMBL3127702)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human histamine H3 receptor expressed in CHOK1 cells after 1.5 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496262(CHEMBL3127683)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496263(CHEMBL3127709)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human histamine H3 receptor expressed in CHOK1 cells after 1.5 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496267(CHEMBL3127686)
Affinity DataIC50: 48nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496275(CHEMBL3127671)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human histamine H3 receptor expressed in CHOK1 cells after 1.5 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496279(CHEMBL3127703)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human histamine H3 receptor expressed in CHOK1 cells after 1.5 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496278(CHEMBL3127706)
Affinity DataIC50: 66nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496268(CHEMBL3127685)
Affinity DataIC50: 66nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496278(CHEMBL3127706)
Affinity DataKi:  67nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human histamine H3 receptor expressed in CHOK1 cells after 1.5 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496279(CHEMBL3127703)
Affinity DataIC50: 74nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496275(CHEMBL3127671)
Affinity DataIC50: 83nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50496259(CHEMBL3127672)
Affinity DataIC50: 87nMAssay Description:Antagonist activity at human histamine H3 receptor long form expressed in CHOK1 cells assessed as inhibition of R-alpha-methylhistamine-induced [35S]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
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