Compile Data Set for Download or QSAR
Report error Found 84 Enz. Inhib. hit(s) with all data for entry = 50043769
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50399165(CHEMBL2180137)
Affinity DataIC50: 189nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446060(CHEMBL3103385)
Affinity DataIC50: 3.44E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446068(CHEMBL3103375)
Affinity DataIC50: 4.55E+3nMAssay Description:Antagonist activity at human P2X1 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM22416(PAROXETINE | CHEMBL490 | (3S,4R)-3-[(1,3-benzodiox...)
Affinity DataIC50: 4.68E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446060(CHEMBL3103385)
Affinity DataIC50: 5.32E+3nMAssay Description:Antagonist activity at human P2X1 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446077(CHEMBL3103401)
Affinity DataIC50: 6.02E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446060(CHEMBL3103385)
Affinity DataIC50: 7.18E+3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446068(CHEMBL3103375)
Affinity DataIC50: 7.78E+3nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446070(CHEMBL3103371)
Affinity DataIC50: 7.98E+3nMAssay Description:Antagonist activity at human P2X3 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446047(Carbamazepine epoxide | Carbatrol)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446063(CHEMBL3103382)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446085(CHEMBL3103367)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM34179(CHEMBL1068 | cid_34312 | Trileptal | SMR000048684 ...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446076(CHEMBL1483754)
Affinity DataIC50: 1.14E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446070(CHEMBL3103371)
Affinity DataIC50: 1.37E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446067(CHEMBL3103377)
Affinity DataIC50: 1.38E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446076(CHEMBL1483754)
Affinity DataIC50: 1.42E+4nMAssay Description:Antagonist activity at human P2X3 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Mouse)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446060(CHEMBL3103385)
Affinity DataIC50: 1.49E+4nMAssay Description:Antagonist activity at mouse P2X4 receptor assessed as inhibition of ATP-induced cytosolic calcium influx preincubated for 30 mins followed by ATP ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446068(CHEMBL3103375)
Affinity DataIC50: 1.52E+4nMAssay Description:Antagonist activity at human P2X3 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446052(CHEMBL3103393)
Affinity DataIC50: 1.53E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446074(CHEMBL3103404)
Affinity DataIC50: 1.92E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446064(CHEMBL3103381)
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50240669(Acetic acid (S)-5-carbamoyl-10,11-dihydro-5H-diben...)
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446070(CHEMBL3103371)
Affinity DataIC50: 2.07E+4nMAssay Description:Antagonist activity at human P2X1 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446081(CHEMBL3103398)
Affinity DataIC50: 2.33E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446076(CHEMBL1483754)
Affinity DataIC50: 2.52E+4nMAssay Description:Antagonist activity at human P2X1 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446073(CHEMBL3103405)
Affinity DataIC50: 2.74E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446072(CHEMBL3103369)
Affinity DataIC50: 2.80E+4nMAssay Description:Antagonist activity at human P2X3 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 3(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446069(CHEMBL3103372)
Affinity DataIC50: 2.98E+4nMAssay Description:Antagonist activity at human P2X3 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446059(CHEMBL3103386)
Affinity DataIC50: 3.06E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446072(CHEMBL3103369)
Affinity DataIC50: 3.38E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446069(CHEMBL3103372)
Affinity DataIC50: 3.41E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446068(CHEMBL3103375)
Affinity DataIC50: 3.59E+4nMAssay Description:Antagonist activity at rat P2X4 receptor assessed as inhibition of ATP-induced calcium influx preincubated for 30 mins followed by ATP addition by Fl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446071(CHEMBL3103370)
Affinity DataIC50: 3.62E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446086(CHEMBL3103366)
Affinity DataIC50: 3.69E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446072(CHEMBL3103369)
Affinity DataIC50: 4.08E+4nMAssay Description:Antagonist activity at human P2X7 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446076(CHEMBL1483754)
Affinity DataIC50: 4.30E+4nMAssay Description:Antagonist activity at rat P2X4 receptor assessed as inhibition of ATP-induced calcium influx preincubated for 30 mins followed by ATP addition by Fl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446053(CHEMBL3103392)
Affinity DataIC50: 5.14E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446058(CHEMBL3103387)
Affinity DataIC50: 5.25E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446060(CHEMBL3103385)
Affinity DataIC50: 5.46E+4nMAssay Description:Antagonist activity at rat P2X4 receptor assessed as inhibition of ATP-induced calcium influx preincubated for 30 mins followed by ATP addition by Fl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446055(CHEMBL3103390)
Affinity DataIC50: 5.46E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446069(CHEMBL3103372)
Affinity DataIC50: 6.88E+4nMAssay Description:Antagonist activity at human P2X1 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446069(CHEMBL3103372)
Affinity DataIC50: 6.93E+4nMAssay Description:Antagonist activity at rat P2X4 receptor assessed as inhibition of ATP-induced calcium influx preincubated for 30 mins followed by ATP addition by Fl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446072(CHEMBL3103369)
Affinity DataIC50: 6.96E+4nMAssay Description:Antagonist activity at human P2X1 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446076(CHEMBL1483754)
Affinity DataIC50: 6.98E+4nMAssay Description:Antagonist activity at human P2X7 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446049(CHEMBL3103395)
Affinity DataIC50: 7.28E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446083(CHEMBL3103402)
Affinity DataIC50: 7.89E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446060(CHEMBL3103385)
Affinity DataIC50: 9.52E+4nMAssay Description:Antagonist activity at human P2X7 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446070(CHEMBL3103371)
Affinity DataIC50: 9.58E+4nMAssay Description:Antagonist activity at rat P2X4 receptor assessed as inhibition of ATP-induced calcium influx preincubated for 30 mins followed by ATP addition by Fl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Mouse)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50446072(CHEMBL3103369)
Affinity DataIC50: 9.84E+4nMAssay Description:Antagonist activity at mouse P2X4 receptor assessed as inhibition of ATP-induced cytosolic calcium influx preincubated for 30 mins followed by ATP ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
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