Compile Data Set for Download or QSAR
Report error Found 61 Enz. Inhib. hit(s) with all data for entry = 50043861
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447515(CHEMBL3115901)
Affinity DataKi:  40nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447528(CHEMBL3115904)
Affinity DataKi:  100nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447516(CHEMBL3115900)
Affinity DataKi:  100nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447515(CHEMBL3115901)
Affinity DataIC50: 130nMAssay Description:Inhibition of human APC using S-2366 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mins by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447523(CHEMBL3115897)
Affinity DataKi:  200nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447516(CHEMBL3115900)
Affinity DataIC50: 260nMAssay Description:Inhibition of human APC using S-2366 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mins by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447514(CHEMBL3115903)
Affinity DataKi:  300nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447521(CHEMBL3115899)
Affinity DataKi:  300nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447515(CHEMBL3115901)
Affinity DataKi:  300nMAssay Description:Competitive inhibition of human coagulation factor 11a using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447517(CHEMBL3115894)
Affinity DataKi:  300nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447522(CHEMBL3115898)
Affinity DataKi:  300nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447525(CHEMBL3115893)
Affinity DataKi:  400nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447528(CHEMBL3115904)
Affinity DataIC50: 470nMAssay Description:Inhibition of human APC using S-2366 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mins by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50193243(({(R)-[2-(4-carbamimidoyl-benzylcarbamoyl)-indan-2...)
Affinity DataKi:  500nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447527(CHEMBL3115905)
Affinity DataKi:  500nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447515(CHEMBL3115901)
Affinity DataIC50: 580nMAssay Description:Inhibition of human coagulation factor 11a using S-2366 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447523(CHEMBL3115897)
Affinity DataIC50: 670nMAssay Description:Inhibition of human APC using S-2366 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mins by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447519(CHEMBL3115906)
Affinity DataKi:  800nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447516(CHEMBL3115900)
Affinity DataKi:  800nMAssay Description:Competitive inhibition of human coagulation factor 11a using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447518(CHEMBL3115892)
Affinity DataKi:  900nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447524(CHEMBL3115896)
Affinity DataKi:  900nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447517(CHEMBL3115894)
Affinity DataIC50: 920nMAssay Description:Inhibition of human APC using S-2366 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mins by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447521(CHEMBL3115899)
Affinity DataIC50: 980nMAssay Description:Inhibition of human APC using S-2366 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mins by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447514(CHEMBL3115903)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human APC using S-2366 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mins by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447522(CHEMBL3115898)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human APC using S-2366 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mins by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447520(CHEMBL3115902)
Affinity DataKi:  1.10E+3nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM29388(Exanta | Melagatran | US11584714, Compound 999 | U...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human APC using S-2366 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mins by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447525(CHEMBL3115893)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human APC using S-2366 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mins by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447527(CHEMBL3115905)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human APC using S-2366 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mins by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447526(CHEMBL3115907)
Affinity DataKi:  1.60E+3nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50193243(({(R)-[2-(4-carbamimidoyl-benzylcarbamoyl)-indan-2...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human APC using S-2366 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mins by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447516(CHEMBL3115900)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human coagulation factor 11a using S-2366 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447519(CHEMBL3115906)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human APC using S-2366 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mins by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447524(CHEMBL3115896)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human APC using S-2366 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mins by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447518(CHEMBL3115892)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human APC using S-2366 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mins by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447520(CHEMBL3115902)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of human APC using S-2366 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mins by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetVitamin K-dependent protein C(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447526(CHEMBL3115907)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human APC using S-2366 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mins by spectrophotom...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447516(CHEMBL3115900)
Affinity DataKi:  8.00E+3nMAssay Description:Competitive inhibition of human coagulation factor 10a using S-2765 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447514(CHEMBL3115903)
Affinity DataKi:  1.40E+4nMAssay Description:Competitive inhibition of human coagulation factor 10a using S-2765 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447515(CHEMBL3115901)
Affinity DataKi: >1.50E+4nMAssay Description:Competitive inhibition of human coagulation factor 10a using S-2765 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50193243(({(R)-[2-(4-carbamimidoyl-benzylcarbamoyl)-indan-2...)
Affinity DataKi:  1.60E+4nMAssay Description:Competitive inhibition of human coagulation factor 10a using S-2765 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447514(CHEMBL3115903)
Affinity DataKi:  1.90E+4nMAssay Description:Competitive inhibition of human coagulation factor 11a using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447518(CHEMBL3115892)
Affinity DataKi: >1.90E+4nMAssay Description:Competitive inhibition of human coagulation factor 11a using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447517(CHEMBL3115894)
Affinity DataKi: >1.90E+4nMAssay Description:Competitive inhibition of human coagulation factor 11a using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50193243(({(R)-[2-(4-carbamimidoyl-benzylcarbamoyl)-indan-2...)
Affinity DataKi: >1.90E+4nMAssay Description:Competitive inhibition of human coagulation factor 11a using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447519(CHEMBL3115906)
Affinity DataKi: >1.90E+4nMAssay Description:Competitive inhibition of human coagulation factor 11a using S-2366 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor XI(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM29388(Exanta | Melagatran | US11584714, Compound 999 | U...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human coagulation factor 11a using S-2366 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM29388(Exanta | Melagatran | US11584714, Compound 999 | U...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of human coagulation factor 10a using S-2765 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447516(CHEMBL3115900)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of human coagulation factor 10a using S-2765 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50447514(CHEMBL3115903)
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of human coagulation factor 10a using S-2765 as substrate preincubated for 300 seconds followed by substrate addition measured after 40 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
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