Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50044155
TargetSerine/threonine-protein kinase B-raf(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50006650(CHEMBL526479)
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50006653(CHEMBL497671)
Affinity DataIC50: 0.220nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50006652(CHEMBL498674)
Affinity DataIC50: 0.340nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50432397(CHEMBL2348989)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50006650(CHEMBL526479)
Affinity DataIC50: 9nMAssay Description:Inhibition of BRAF (unknown origin)-mediated ERK phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50006651(CHEMBL3133758)
Affinity DataIC50: 22nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50432397(CHEMBL2348989)
Affinity DataIC50: 43nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50006651(CHEMBL3133758)
Affinity DataIC50: 95nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50006651(CHEMBL3133758)
Affinity DataIC50: 165nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50006649(CHEMBL3235904)
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of N-terminal 6X-His tagged human wild-type BRAF by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed