Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50043893
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50448075(CHEMBL1258979)
Affinity DataIC50: 9.91E+3nMAssay Description:Inverse agonist activity at human GPR18 expressed in CHO cells assessed as inhibition of 7.5 uM THC-mediated beta-arrestin recruitment after 90 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50448074(Emindole Sb)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR55 expressed in CHO cells assessed as inhibition of LPI-mediated beta-arrestin recruitment after 90 mins by beta-gala...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50448074(Emindole Sb)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR18 expressed in CHO cells assessed as inhibition of 10 uM THC-mediated beta-arrestin recruitment after 90 mins by bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50448073(CHEMBL3120631)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR18 expressed in CHO cells assessed as inhibition of 10 uM THC-mediated beta-arrestin recruitment after 90 mins by bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50448073(CHEMBL3120631)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR55 expressed in CHO cells assessed as inhibition of LPI-mediated beta-arrestin recruitment after 90 mins by beta-gala...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50448076(CHEMBL3120632)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR55 expressed in CHO cells assessed as inhibition of LPI-mediated beta-arrestin recruitment after 90 mins by beta-gala...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50448075(CHEMBL1258979)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR55 expressed in CHO cells assessed as inhibition of LPI-mediated beta-arrestin recruitment after 90 mins by beta-gala...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetN-arachidonyl glycine receptor(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50448076(CHEMBL3120632)
Affinity DataIC50: 1.34E+4nMAssay Description:Inverse agonist activity at human GPR18 expressed in CHO cells assessed as inhibition of 7.5 uM THC-mediated beta-arrestin recruitment after 90 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed