Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50043821
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50446727(CHEMBL3114111)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50446726(CHEMBL3114112)
Affinity DataIC50: 1.20E+3nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50446733(CHEMBL3114123)
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50446725(CHEMBL3114113)
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50446723(CHEMBL3114115)
Affinity DataIC50: 2.90E+3nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50446716(CHEMBL3114120)
Affinity DataIC50: 3.10E+3nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50446721(CHEMBL1205188)
Affinity DataIC50: 3.10E+3nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50446732(CHEMBL3114124)
Affinity DataIC50: 3.20E+3nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50446724(CHEMBL3114114)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50446731(CHEMBL3114125)
Affinity DataIC50: 3.50E+3nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50446718(CHEMBL3114118)
Affinity DataIC50: 5.40E+3nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50446728(CHEMBL3114110)
Affinity DataIC50: 5.50E+3nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50446734(CHEMBL3114122)
Affinity DataIC50: 5.80E+3nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50446729(CHEMBL3114109)
Affinity DataIC50: 7.80E+3nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50446717(CHEMBL3114119)
Affinity DataIC50: 8.40E+3nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50446720(CHEMBL3114116)
Affinity DataIC50: 8.50E+3nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50446719(CHEMBL3114117)
Affinity DataIC50: 8.60E+3nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50446730(CHEMBL3114126)
Affinity DataIC50: 8.70E+3nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50446735(CHEMBL3114121)
Affinity DataIC50: 2.52E+4nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM81519(LY 255283 | CHEMBL15766 | CAS_117690-79-6 | CGS 23...)
Affinity DataIC50: 3.52E+4nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM21725((1S,2R,10R,11S,14Z,15S)-14-ethylidene-2,15-dimethy...)
Affinity DataIC50: 8.94E+4nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBile acid receptor(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50446722(CHEMBL53417)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at GST-tagged FXRalpha LBD (unknown origin) assessed as inhibition of CDCA-induced bio-SRC-1 recruitment after 30 mins by fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed