Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50043912
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448377(CHEMBL3121473)
Affinity DataEC50:  0.0794nMAssay Description:Agonist activity at muscarinic M2 receptor in albino guinea pig left atrium assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448377(CHEMBL3121473)
Affinity DataEC50:  0.166nMAssay Description:Agonist activity at muscarinic M3 receptor in albino guinea pig ileum assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448375(CHEMBL3121479)
Affinity DataEC50:  7.10nMAssay Description:Agonist activity at muscarinic M2 receptor in albino guinea pig left atrium assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448374(CHEMBL3121478)
Affinity DataEC50:  7.80nMAssay Description:Agonist activity at muscarinic M2 receptor in albino guinea pig left atrium assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448375(CHEMBL3121479)
Affinity DataEC50:  11nMAssay Description:Agonist activity at muscarinic M3 receptor in albino guinea pig ileum assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448372(CHEMBL3121475)
Affinity DataEC50:  12nMAssay Description:Agonist activity at muscarinic M2 receptor in albino guinea pig left atrium assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448369(CHEMBL3121476)
Affinity DataEC50:  14nMAssay Description:Agonist activity at muscarinic M2 receptor in albino guinea pig left atrium assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448370(CHEMBL3120178)
Affinity DataEC50:  19nMAssay Description:Agonist activity at muscarinic M2 receptor in albino guinea pig left atrium assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448374(CHEMBL3121478)
Affinity DataEC50:  21nMAssay Description:Agonist activity at muscarinic M3 receptor in albino guinea pig ileum assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448371(CHEMBL3121480)
Affinity DataEC50:  21nMAssay Description:Agonist activity at muscarinic M2 receptor in albino guinea pig left atrium assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448373(CHEMBL3121477)
Affinity DataEC50:  38nMAssay Description:Agonist activity at muscarinic M2 receptor in albino guinea pig left atrium assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448371(CHEMBL3121480)
Affinity DataEC50:  47nMAssay Description:Agonist activity at muscarinic M3 receptor in albino guinea pig ileum assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448370(CHEMBL3120178)
Affinity DataEC50:  50nMAssay Description:Agonist activity at muscarinic M3 receptor in albino guinea pig ileum assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448378(CHEMBL3121474)
Affinity DataEC50:  66nMAssay Description:Agonist activity at muscarinic M2 receptor in albino guinea pig left atrium assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448369(CHEMBL3121476)
Affinity DataEC50:  69nMAssay Description:Agonist activity at muscarinic M3 receptor in albino guinea pig ileum assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448373(CHEMBL3121477)
Affinity DataEC50:  69nMAssay Description:Agonist activity at muscarinic M3 receptor in albino guinea pig ileum assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448372(CHEMBL3121475)
Affinity DataEC50:  105nMAssay Description:Agonist activity at muscarinic M3 receptor in albino guinea pig ileum assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448378(CHEMBL3121474)
Affinity DataEC50:  871nMAssay Description:Agonist activity at muscarinic M3 receptor in albino guinea pig ileum assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandPNGBDBM39342(2-carbamoyloxypropyl(trimethyl)azanium;chloride | ...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at muscarinic M3 receptor in albino guinea pig ileum assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Milan

Curated by ChEMBL
LigandPNGBDBM39342(2-carbamoyloxypropyl(trimethyl)azanium;chloride | ...)
Affinity DataEC50:  1.41E+3nMAssay Description:Agonist activity at muscarinic M2 receptor in albino guinea pig left atrium assessed as stimulation of electrically-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetAcetylcholine receptor subunit epsilon(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448370(CHEMBL3120178)
Affinity DataIC50: 7.94E+3nMAssay Description:Inhibition of acetylcholinesterase in rat brain homogenate after 15 mins by Ellman assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetAcetylcholine receptor subunit epsilon(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448375(CHEMBL3121479)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of acetylcholinesterase in rat brain homogenate after 15 mins by Ellman assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetAcetylcholine receptor subunit epsilon(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448374(CHEMBL3121478)
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of acetylcholinesterase in rat brain homogenate after 15 mins by Ellman assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetAcetylcholine receptor subunit epsilon(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448369(CHEMBL3121476)
Affinity DataIC50: 1.95E+4nMAssay Description:Inhibition of acetylcholinesterase in rat brain homogenate after 15 mins by Ellman assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetAcetylcholine receptor subunit epsilon(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448371(CHEMBL3121480)
Affinity DataIC50: 2.29E+4nMAssay Description:Inhibition of acetylcholinesterase in rat brain homogenate after 15 mins by Ellman assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetAcetylcholine receptor subunit epsilon(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448372(CHEMBL3121475)
Affinity DataIC50: 3.16E+4nMAssay Description:Inhibition of acetylcholinesterase in rat brain homogenate after 15 mins by Ellman assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetAcetylcholine receptor subunit epsilon(Rat)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50448376(Naphmethonium)
Affinity DataIC50: 4.17E+4nMAssay Description:Inhibition of acetylcholinesterase in rat brain homogenate after 15 mins by Ellman assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed