Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50043979
TargetTyrosine-protein kinase SYK(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM92625(Dimethoxyquinoline, 2)
Affinity DataIC50: 100nMAssay Description:Inhibition of Syk (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein kinase JAK2(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50449315(CHEMBL3125863)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50449315(CHEMBL3125863)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of ZAP70 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetTyrosine-protein kinase ZAP-70(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50449314(CHEMBL3125862)
Affinity DataIC50: 8.60E+3nMAssay Description:Inhibition of ZAP70 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50449314(CHEMBL3125862)
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of JAK2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50449315(CHEMBL3125863)
Affinity DataIC50: 1.84E+4nMAssay Description:Inhibition of Syk (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50449314(CHEMBL3125862)
Affinity DataIC50: 2.26E+4nMAssay Description:Inhibition of Syk (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50449315(CHEMBL3125863)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of c-MET (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50449314(CHEMBL3125862)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of c-MET (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50449315(CHEMBL3125863)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of FAK (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
University of Zurich

Curated by ChEMBL
LigandPNGBDBM50449314(CHEMBL3125862)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of FAK (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed