Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50044117
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50216689(2-cyano-3-(5-(2,5-dichlorophenyl)furan-2-yl)-N-(qu...)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human recombinant SIRT2 using Fluor-de-Lys as substrate incubated for 60 mins prior to substrate addition measured after 60 mins by flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50004135(CHEMBL3236132)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of human recombinant SIRT2 using Fluor-de-Lys as substrate incubated for 60 mins prior to substrate addition measured after 60 mins by flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50004137(CHEMBL3236133)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of human recombinant SIRT2 using Fluor-de-Lys as substrate incubated for 60 mins prior to substrate addition measured after 60 mins by flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50216689(2-cyano-3-(5-(2,5-dichlorophenyl)furan-2-yl)-N-(qu...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human recombinant SIRT1 using Fluor-de-Lys as substrate incubated for 60 mins prior to substrate addition measured after 60 mins by flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50216689(2-cyano-3-(5-(2,5-dichlorophenyl)furan-2-yl)-N-(qu...)
Affinity DataIC50: 9.10E+4nMAssay Description:Inhibition of human recombinant SIRT3 using Fluor-de-Lys as substrate incubated for 60 mins prior to substrate addition measured after 60 mins by flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50004135(CHEMBL3236132)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant SIRT3 using Fluor-de-Lys as substrate incubated for 60 mins prior to substrate addition measured after 60 mins by flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50004137(CHEMBL3236133)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant SIRT3 using Fluor-de-Lys as substrate incubated for 60 mins prior to substrate addition measured after 60 mins by flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50004137(CHEMBL3236133)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant SIRT1 using Fluor-de-Lys as substrate incubated for 60 mins prior to substrate addition measured after 60 mins by flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50004135(CHEMBL3236132)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant SIRT1 using Fluor-de-Lys as substrate incubated for 60 mins prior to substrate addition measured after 60 mins by flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed