Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50006104
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50103642(CHEMBL308954 | TMC-125 | TMC 125 | 4-(6-amino-5-br...)
Affinity DataIC50: 16nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase p66/p51 after 40 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM2483(Sustiva | DMP-266 | (4S)-6-chloro-4-(2-cyclopropyl...)
Affinity DataIC50: 38nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase p66/p51 after 40 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50496958(CHEMBL3236843)
Affinity DataIC50: 160nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase p66/p51 after 40 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50496955(CHEMBL3236849)
Affinity DataIC50: 390nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase p66/p51 after 40 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50496956(CHEMBL3236847)
Affinity DataIC50: 630nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase p66/p51 after 40 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM1434(BI-RG-587 | 2-cyclopropyl-7-methyl-2,4,9,15-tetraa...)
Affinity DataIC50: 1.78E+3nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase p66/p51 after 40 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50496957(CHEMBL3236842)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptase p66/p51 after 40 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed