Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 6343
TargetProteasome subunit beta type-5(Human)
Zhejiang University

LigandPNGBDBM50277889(CHEMBL451887 | CARFILZOMIB)
Affinity DataIC50: 8.60nMAssay Description:The assay was carried out in 50 uL volume, where 1 uL compound was added to 10 uL purified human proteasome (25 ug/mL) and incubated for 15 min and t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Zhejiang University

LigandPNGBDBM50069989(CHEMBL325041 | (R)-3-methyl-1-((S)-3-phenyl-2-(pyr...)
Affinity DataIC50: 8.96nMAssay Description:The assay was carried out in 50 uL volume, where 1 uL compound was added to 10 uL purified human proteasome (25 ug/mL) and incubated for 15 min and t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Zhejiang University

LigandPNGBDBM123812(4-Fluoro-N-{3-{S-4-methyl-1-[S-4-methyl-1-(R-2-met...)
Affinity DataIC50: 970nMAssay Description:The assay was carried out in 50 uL volume, where 1 uL compound was added to 10 uL purified human proteasome (25 ug/mL) and incubated for 15 min and t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Zhejiang University

LigandPNGBDBM123813(4-Methoxy-N-{3-{S-4-methyl-1-[S-4-methyl-1-(R-2-me...)
Affinity DataIC50: 1.01E+3nMAssay Description:The assay was carried out in 50 uL volume, where 1 uL compound was added to 10 uL purified human proteasome (25 ug/mL) and incubated for 15 min and t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Zhejiang University

LigandPNGBDBM123811(N-{3-{S-4-Methyl-1-[S-4-methyl-1-(R-2-methyloxiran...)
Affinity DataIC50: 1.42E+3nMAssay Description:The assay was carried out in 50 uL volume, where 1 uL compound was added to 10 uL purified human proteasome (25 ug/mL) and incubated for 15 min and t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Zhejiang University

LigandPNGBDBM123810(N-{3-{S-4-Methyl-1-[S-4-methyl-1-(R-2-methyloxiran...)
Affinity DataIC50: 1.85E+3nMAssay Description:The assay was carried out in 50 uL volume, where 1 uL compound was added to 10 uL purified human proteasome (25 ug/mL) and incubated for 15 min and t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details Article
PubMed