Compile Data Set for Download or QSAR
Report error Found 59 Enz. Inhib. hit(s) with all data for entry = 50044387
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015421(CHEMBL3264644)
Affinity DataIC50: 7.5nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015419(CHEMBL3264642)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015403(CHEMBL3264636)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015405(CHEMBL3264637)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50236238(5beta-cholanic acid-3alpha-ol | CHEMBL1478 | (3alp...)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015382(CHEMBL3264645)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015414(CHEMBL3264639)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM21724(3-[(E)-2-(2-chloro-4-{[3-(2,6-dichlorophenyl)-5-(p...)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015402(CHEMBL3264635)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015412(CHEMBL3264638)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015388(CHEMBL3264651)
Affinity DataIC50: 31nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015386(CHEMBL3264649)
Affinity DataIC50: 43nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015401(CHEMBL1367639)
Affinity DataIC50: 47nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015417(CHEMBL3264640)
Affinity DataIC50: 49nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015418(CHEMBL3264641)
Affinity DataIC50: 53nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015420(CHEMBL3264643)
Affinity DataIC50: 77nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015387(CHEMBL3264650)
Affinity DataIC50: 78nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015383(CHEMBL3264646)
Affinity DataIC50: 130nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015385(CHEMBL3264648)
Affinity DataIC50: 160nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015384(CHEMBL3264647)
Affinity DataIC50: 199nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015390(CHEMBL3264987)
Affinity DataIC50: 390nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015421(CHEMBL3264644)
Affinity DataIC50: 469nMAssay Description:Inhibition of GW4064-induced transactivation of FXR (unknown origin) expressed in HEK293T cells after 16 hrs by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015391(CHEMBL3264988)
Affinity DataIC50: 489nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015382(CHEMBL3264645)
Affinity DataIC50: 515nMAssay Description:Inhibition of GW4064-induced transactivation of FXR (unknown origin) expressed in HEK293T cells after 16 hrs by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015388(CHEMBL3264651)
Affinity DataIC50: 593nMAssay Description:Inhibition of GW4064-induced transactivation of FXR (unknown origin) expressed in HEK293T cells after 16 hrs by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015419(CHEMBL3264642)
Affinity DataIC50: 844nMAssay Description:Inhibition of GW4064-induced transactivation of FXR (unknown origin) expressed in HEK293T cells after 16 hrs by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015420(CHEMBL3264643)
Affinity DataIC50: 849nMAssay Description:Inhibition of GW4064-induced transactivation of FXR (unknown origin) expressed in HEK293T cells after 16 hrs by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015398(CHEMBL3264627)
Affinity DataIC50: 996nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015386(CHEMBL3264649)
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibition of GW4064-induced transactivation of FXR (unknown origin) expressed in HEK293T cells after 16 hrs by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015405(CHEMBL3264637)
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibition of GW4064-induced transactivation of FXR (unknown origin) expressed in HEK293T cells after 16 hrs by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015399(CHEMBL3264629)
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015417(CHEMBL3264640)
Affinity DataIC50: 1.69E+3nMAssay Description:Inhibition of GW4064-induced transactivation of FXR (unknown origin) expressed in HEK293T cells after 16 hrs by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015387(CHEMBL3264650)
Affinity DataIC50: 1.95E+3nMAssay Description:Inhibition of GW4064-induced transactivation of FXR (unknown origin) expressed in HEK293T cells after 16 hrs by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015394(CHEMBL3264991)
Affinity DataIC50: 2.04E+3nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015395(CHEMBL3264992)
Affinity DataIC50: 2.31E+3nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015402(CHEMBL3264635)
Affinity DataIC50: 2.49E+3nMAssay Description:Inhibition of GW4064-induced transactivation of FXR (unknown origin) expressed in HEK293T cells after 16 hrs by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015383(CHEMBL3264646)
Affinity DataIC50: 2.61E+3nMAssay Description:Inhibition of GW4064-induced transactivation of FXR (unknown origin) expressed in HEK293T cells after 16 hrs by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015401(CHEMBL1367639)
Affinity DataIC50: 2.62E+3nMAssay Description:Inhibition of GW4064-induced transactivation of FXR (unknown origin) expressed in HEK293T cells after 16 hrs by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015384(CHEMBL3264647)
Affinity DataIC50: 3.11E+3nMAssay Description:Inhibition of GW4064-induced transactivation of FXR (unknown origin) expressed in HEK293T cells after 16 hrs by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015396(CHEMBL3264624)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015389(CHEMBL3264652)
Affinity DataIC50: 3.42E+3nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015385(CHEMBL3264648)
Affinity DataIC50: 3.49E+3nMAssay Description:Inhibition of GW4064-induced transactivation of FXR (unknown origin) expressed in HEK293T cells after 16 hrs by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015393(CHEMBL3264990)
Affinity DataIC50: 3.81E+3nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015392(CHEMBL3264989)
Affinity DataIC50: 5.33E+3nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015403(CHEMBL3264636)
Affinity DataIC50: 5.91E+3nMAssay Description:Inhibition of GW4064-induced transactivation of FXR (unknown origin) expressed in HEK293T cells after 16 hrs by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015400(CHEMBL3264630)
Affinity DataIC50: 6.60E+3nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015414(CHEMBL3264639)
Affinity DataIC50: 7.91E+3nMAssay Description:Inhibition of GW4064-induced transactivation of FXR (unknown origin) expressed in HEK293T cells after 16 hrs by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015397(CHEMBL3264626)
Affinity DataIC50: 8.30E+3nMAssay Description:Antagonist activity at human GST-tagged FXR after 20 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015397(CHEMBL3264626)
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of GW4064-induced transactivation of FXR (unknown origin) expressed in HEK293T cells after 16 hrs by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Beckman Research Institute

Curated by ChEMBL
LigandPNGBDBM50015399(CHEMBL3264629)
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of GW4064-induced transactivation of FXR (unknown origin) expressed in HEK293T cells after 16 hrs by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
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