Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50044506
TargetMuscarinic acetylcholine receptor M4(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50019336(CHEMBL3289442)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human muscarinic acetylcholine receptor M4 expressed in CHO cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50019335(CHEMBL3289440)
Affinity DataEC50:  93nMAssay Description:Agonist activity at human muscarinic acetylcholine receptor M4 expressed in CHO cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50019335(CHEMBL3289440)
Affinity DataEC50:  352nMAssay Description:Agonist activity at human muscarinic acetylcholine receptor M1 expressed in CHO cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50019335(CHEMBL3289440)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human ERG tail current after 5 mins by patch-clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50019334(CHEMBL3289444)
Affinity DataIC50: 2.75E+3nMAssay Description:Inhibition of human ERG tail current after 5 mins by patch-clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50019336(CHEMBL3289442)
Affinity DataIC50: 3.63E+3nMAssay Description:Inhibition of human ERG tail current after 5 mins by patch-clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50019337(CHEMBL3289443)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human ERG tail current after 5 mins by patch-clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed