Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50044506
Affinity DataEC50: 13nMAssay Description:Agonist activity at human muscarinic acetylcholine receptor M4 expressed in CHO cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 93nMAssay Description:Agonist activity at human muscarinic acetylcholine receptor M4 expressed in CHO cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 352nMAssay Description:Agonist activity at human muscarinic acetylcholine receptor M1 expressed in CHO cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human ERG tail current after 5 mins by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 2.75E+3nMAssay Description:Inhibition of human ERG tail current after 5 mins by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 3.63E+3nMAssay Description:Inhibition of human ERG tail current after 5 mins by patch-clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Dainippon Sumitomo Pharma
Curated by ChEMBL
Dainippon Sumitomo Pharma
Curated by ChEMBL
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human ERG tail current after 5 mins by patch-clamp methodMore data for this Ligand-Target Pair



