Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50044512
TargetSerine/threonine-protein kinase B-raf(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataIC50: 120nMAssay Description:Binding affinity to B-RAF kinase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase B-raf(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataIC50: 136nMAssay Description:Competitive binding affinity to B-RAF kinase (unknown origin) after 60 to 120 mins by FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019448(CHEMBL3290437)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019432(CHEMBL3290698)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019436(CHEMBL3290699)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019437(CHEMBL3290430)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019441(CHEMBL3290431)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019442(CHEMBL3290432)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019444(CHEMBL3290433)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019445(CHEMBL3290434)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019446(CHEMBL3290435)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019447(CHEMBL3290436)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019429(CHEMBL3290697)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019449(CHEMBL3290438)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019450(CHEMBL3290687)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019451(CHEMBL3290688)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019452(CHEMBL3290689)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019453(CHEMBL3290690)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019454(CHEMBL3290691)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019455(CHEMBL3290692)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019456(CHEMBL3290693)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019459(CHEMBL3290694)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019460(CHEMBL3290695)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019449(CHEMBL3290438)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019429(CHEMBL3290697)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019432(CHEMBL3290698)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019436(CHEMBL3290699)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019437(CHEMBL3290430)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019441(CHEMBL3290431)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019442(CHEMBL3290432)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019444(CHEMBL3290433)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019445(CHEMBL3290434)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019446(CHEMBL3290435)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019447(CHEMBL3290436)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019448(CHEMBL3290437)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019428(CHEMBL3290696)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant casein kinase-1 delta using casein as substrate after 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019450(CHEMBL3290687)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019451(CHEMBL3290688)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019452(CHEMBL3290689)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019453(CHEMBL3290690)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019454(CHEMBL3290691)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019455(CHEMBL3290692)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019456(CHEMBL3290693)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019459(CHEMBL3290694)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019460(CHEMBL3290695)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Trinity College

Curated by ChEMBL
LigandPNGBDBM50019428(CHEMBL3290696)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant GSK-3 beta after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed