Compile Data Set for Download or QSAR
Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 50033065
LigandPNGBDBM50339043(2-(2-((4-Pyridyl)methyl)aminophenyl)-5-(3,4-ethyle...)
Affinity DataIC50: 110nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339053(N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-5-(2-(quin...)
Affinity DataIC50: 150nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339046(5-(2-((1H-imidazol-5-yl)methylamino)pyridin-3-yl)-...)
Affinity DataIC50: 160nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50179492(3-(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-ylamino)-1,...)
Affinity DataIC50: 170nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339043(2-(2-((4-Pyridyl)methyl)aminophenyl)-5-(3,4-ethyle...)
Affinity DataIC50: 210nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339048(N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-5-(2-(quin...)
Affinity DataIC50: 220nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339048(N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-5-(2-(quin...)
Affinity DataIC50: 300nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339046(5-(2-((1H-imidazol-5-yl)methylamino)pyridin-3-yl)-...)
Affinity DataIC50: 830nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339054(2-(2-((4-Pyridyl)methyl)aminophenyl)-5-(3,4-methyl...)
Affinity DataIC50: 830nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339037(N-(pyridin-4-ylmethyl)-3-(5-(3-(trifluoromethyl)ph...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50179492(3-(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-ylamino)-1,...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339037(N-(pyridin-4-ylmethyl)-3-(5-(3-(trifluoromethyl)ph...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339047(5-(2-((1H-indazol-5-yl)methylamino)pyridin-3-yl)-N...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50179495(3-(5-(benzo[d][1,3]dioxol-5-ylamino)-1,3,4-oxadiaz...)
Affinity DataIC50: 1.89E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339040(3-(5-(benzo[d][1,3]dioxol-5-yl)-4H-1,2,4-triazol-3...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339039(N-(pyridin-4-ylmethyl)-3-(5-(3-(trifluoromethyl)ph...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50179502(N-(benzo[d][1,3]dioxol-5-ylmethyl)-3-(5-(2,3-dihyd...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339050(N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-5-(2-(pyri...)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339052(5-(2-((1H-indazol-5-yl)methylamino)phenyl)-N-(2,3-...)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339055(N-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)-5-(2-(pyr...)
Affinity DataIC50: 3.16E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339050(N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-5-(2-(pyri...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339057(N-(benzo[d][1,3]dioxol-5-yl)-5-(2-(2-(pyridin-3-yl...)
Affinity DataIC50: 3.41E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339041(N-((1,4-dioxan-2-yl)methyl)-3-(5-(4-(methylsulfony...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339051(5-(2-((1H-imidazol-5-yl)methylamino)phenyl)-N-(2,3...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339049(N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-5-(2-(pyri...)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339052(5-(2-((1H-indazol-5-yl)methylamino)phenyl)-N-(2,3-...)
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339053(N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-5-(2-(quin...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339051(5-(2-((1H-imidazol-5-yl)methylamino)phenyl)-N-(2,3...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339049(N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-5-(2-(pyri...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50179487(3-(5-(benzo[d][1,3]dioxol-5-ylamino)-1,3,4-oxadiaz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50179498(3-(5-(benzo[d][1,3]dioxol-5-ylamino)-1,3,4-oxadiaz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339047(5-(2-((1H-indazol-5-yl)methylamino)pyridin-3-yl)-N...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339056(N-(benzo[d][1,3]dioxol-5-yl)-5-(2-(benzo[d][1,3]di...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339045(N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-5-(2-(2-(p...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339044(N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-5-(2-(2-(p...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50179502(N-(benzo[d][1,3]dioxol-5-ylmethyl)-3-(5-(2,3-dihyd...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339055(N-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)-5-(2-(pyr...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339041(N-((1,4-dioxan-2-yl)methyl)-3-(5-(4-(methylsulfony...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339038(N-((1H-pyrazol-4-yl)methyl)-3-(5-(3-(trifluorometh...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339042(N-(benzo[d][1,3]dioxol-5-yl)-5-(2-(2-(pyridin-4-yl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50179501(3-(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-ylamino)-1,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50179504(3-(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-ylamino)-1,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339044(N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-5-(2-(2-(p...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339045(N-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-5-(2-(2-(p...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR-2 kinase assessed as phosphorylated level of pGAT-biotin peptide preincubated for 5 to 10 mins before addition of substrate measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339038(N-((1H-pyrazol-4-yl)methyl)-3-(5-(3-(trifluorometh...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339039(N-(pyridin-4-ylmethyl)-3-(5-(3-(trifluoromethyl)ph...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339040(3-(5-(benzo[d][1,3]dioxol-5-yl)-4H-1,2,4-triazol-3...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50179504(3-(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-ylamino)-1,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50179495(3-(5-(benzo[d][1,3]dioxol-5-ylamino)-1,3,4-oxadiaz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50339054(2-(2-((4-Pyridyl)methyl)aminophenyl)-5-(3,4-methyl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of VEGFR2 expressed HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
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