Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50043503
TargetAndrogen receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM35909(Eulexin | 2-hydroxy-2-methyl-N-(4-nitro-3-(trifluo...)
Affinity DataIC50: 370nMAssay Description:Antagonist activity at androgen receptor in mouse SC3 cells assessed as inhibition of DHT-induced cell growth after 3 days by CCK-8/WST-8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442124(CHEMBL2441094)
Affinity DataIC50: 750nMAssay Description:Antagonist activity at androgen receptor in mouse SC3 cells assessed as inhibition of DHT-induced cell growth after 3 days by CCK-8/WST-8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442125(CHEMBL2441107)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at androgen receptor in mouse SC3 cells assessed as inhibition of DHT-induced cell growth after 3 days by CCK-8/WST-8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442123(CHEMBL2441092)
Affinity DataIC50: 2.90E+3nMAssay Description:Antagonist activity at androgen receptor in mouse SC3 cells assessed as inhibition of DHT-induced cell growth after 3 days by CCK-8/WST-8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442131(CHEMBL2441100)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at androgen receptor in mouse SC3 cells assessed as inhibition of DHT-induced cell growth after 3 days by CCK-8/WST-8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442123(CHEMBL2441092)
Affinity DataIC50: 5.40E+3nMAssay Description:Displacement of [3H]-DHT from human GST-tagged androgen receptor LBD (627 to 919) expressed in Escherichia coli HB-101 after 15 hrs by liquid scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442121(CHEMBL2441091)
Affinity DataIC50: 5.90E+3nMAssay Description:Antagonist activity at androgen receptor in mouse SC3 cells assessed as inhibition of DHT-induced cell growth after 3 days by CCK-8/WST-8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442130(CHEMBL2441098)
Affinity DataIC50: 6.70E+3nMAssay Description:Antagonist activity at androgen receptor in mouse SC3 cells assessed as inhibition of DHT-induced cell growth after 3 days by CCK-8/WST-8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM35909(Eulexin | 2-hydroxy-2-methyl-N-(4-nitro-3-(trifluo...)
Affinity DataIC50: 7.10E+3nMAssay Description:Displacement of [3H]-DHT from human GST-tagged androgen receptor LBD (627 to 919) expressed in Escherichia coli HB-101 after 15 hrs by liquid scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442122(CHEMBL2441093)
Affinity DataIC50: 7.20E+3nMAssay Description:Antagonist activity at androgen receptor in mouse SC3 cells assessed as inhibition of DHT-induced cell growth after 3 days by CCK-8/WST-8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442129(CHEMBL2441099)
Affinity DataIC50: 8.70E+3nMAssay Description:Antagonist activity at androgen receptor in mouse SC3 cells assessed as inhibition of DHT-induced cell growth after 3 days by CCK-8/WST-8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442135(CHEMBL2441105)
Affinity DataIC50: 8.80E+3nMAssay Description:Antagonist activity at androgen receptor in mouse SC3 cells assessed as inhibition of DHT-induced cell growth after 3 days by CCK-8/WST-8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442124(CHEMBL2441094)
Affinity DataIC50: 9.20E+3nMAssay Description:Displacement of [3H]-DHT from human GST-tagged androgen receptor LBD (627 to 919) expressed in Escherichia coli HB-101 after 15 hrs by liquid scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442138(CHEMBL2441110)
Affinity DataIC50: 9.40E+3nMAssay Description:Antagonist activity at androgen receptor in mouse SC3 cells assessed as inhibition of DHT-induced cell growth after 3 days by CCK-8/WST-8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442128(CHEMBL2441097)
Affinity DataIC50: 9.70E+3nMAssay Description:Antagonist activity at androgen receptor in mouse SC3 cells assessed as inhibition of DHT-induced cell growth after 3 days by CCK-8/WST-8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442121(CHEMBL2441091)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]-DHT from human GST-tagged androgen receptor LBD (627 to 919) expressed in Escherichia coli HB-101 after 15 hrs by liquid scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442132(CHEMBL2441101)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at androgen receptor in mouse SC3 cells assessed as inhibition of DHT-induced cell growth after 3 days by CCK-8/WST-8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442133(CHEMBL2441103)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at androgen receptor in mouse SC3 cells assessed as inhibition of DHT-induced cell growth after 3 days by CCK-8/WST-8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442134(CHEMBL2441102)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at androgen receptor in mouse SC3 cells assessed as inhibition of DHT-induced cell growth after 3 days by CCK-8/WST-8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442127(CHEMBL2441095)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at androgen receptor in mouse SC3 cells assessed as inhibition of DHT-induced cell growth after 3 days by CCK-8/WST-8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442136(CHEMBL2441108)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at androgen receptor in mouse SC3 cells assessed as inhibition of DHT-induced cell growth after 3 days by CCK-8/WST-8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442126(CHEMBL2441096)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at androgen receptor in mouse SC3 cells assessed as inhibition of DHT-induced cell growth after 3 days by CCK-8/WST-8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442137(CHEMBL2441109)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at androgen receptor in mouse SC3 cells assessed as inhibition of DHT-induced cell growth after 3 days by CCK-8/WST-8 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442122(CHEMBL2441093)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]-DHT from human GST-tagged androgen receptor LBD (627 to 919) expressed in Escherichia coli HB-101 after 15 hrs by liquid scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442125(CHEMBL2441107)
Affinity DataIC50: 2.00E+4nMAssay Description:Displacement of [3H]-DHT from human GST-tagged androgen receptor LBD (627 to 919) expressed in Escherichia coli HB-101 after 15 hrs by liquid scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed