Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50005259
TargetTranscription factor 7-like 2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50014132(CHEMBL2323032)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetTranscription factor 7-like 2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM32102(cid_66541 | 1,6-dimethylpyrimido[5,4-e][1,2,4]tria...)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetTranscription factor 7-like 2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50014132(CHEMBL2323032)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetTranscription factor 7-like 2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM32102(cid_66541 | 1,6-dimethylpyrimido[5,4-e][1,2,4]tria...)
Affinity DataKi:  5.80E+3nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetTranscription factor 7-like 2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50094484(CHEMBL2323033 | CHEBI:3556 | US9284299, CGP049090 ...)
Affinity DataKi:  5.90E+3nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetTranscription factor 7-like 2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50094600(CHEMBL2323029)
Affinity DataKi:  8.80E+3nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetTranscription factor 7-like 2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50094600(CHEMBL2323029)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetTranscription factor 7-like 2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50489463(CHEMBL2323031)
Affinity DataKi:  1.60E+4nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetTranscription factor 7-like 2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50249236(CHEMBL460433 | (R)-1-(4,9-dihydroxy-12-((R)-2-((4-...)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetTranscription factor 7-like 2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50094597(CHEMBL2323028)
Affinity DataKi:  2.10E+4nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetTranscription factor 7-like 2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50489463(CHEMBL2323031)
Affinity DataKi:  2.10E+4nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetTranscription factor 7-like 2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50489464(CHEMBL2323030)
Affinity DataKi:  2.90E+4nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetTranscription factor 7-like 2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50094484(CHEMBL2323033 | CHEBI:3556 | US9284299, CGP049090 ...)
Affinity DataKi:  3.60E+4nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetTranscription factor 7-like 2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50094597(CHEMBL2323028)
Affinity DataKi:  7.70E+4nMAssay Description:Inhibition of human beta-casein/Tcf4 interaction after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed