Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 50042590
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428265(CHEMBL2337020)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428256(CHEMBL2337027)
Affinity DataKd:  2.20E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428257(CHEMBL2337026)
Affinity DataKd:  3.50E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428258(CHEMBL2337025)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428259(CHEMBL2331612)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428260(CHEMBL2337024)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428261(CHEMBL2337023)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428262(CHEMBL2337022)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428263(CHEMBL2337021)
Affinity DataKd:  6.60E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428264(CHEMBL1559278)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428254(CHEMBL1609857)
Affinity DataKd:  7.00E+3nMAssay Description:Displacement of MLL-WIN N-terminal FITC-tagged GSARAEVHLRKS peptide from human WDR5 (1-334) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428266(CHEMBL2337019)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428267(CHEMBL2337018)
Affinity DataKd:  1.50E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428268(CHEMBL2337017)
Affinity DataKd:  710nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428269(CHEMBL2337016)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428270(CHEMBL1407785)
Affinity DataKd:  5.80E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428271(CHEMBL2337032)
Affinity DataKd:  270nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428272(CHEMBL2337031)
Affinity DataKd:  680nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428273(CHEMBL2337030)
Affinity DataKd:  590nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428274(CHEMBL2337029)
Affinity DataKd:  630nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428246(CHEMBL2337441)
Affinity DataKd: >2.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428236(CHEMBL1457864)
Affinity DataKd:  1.40E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428237(CHEMBL2337450)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428238(CHEMBL2337449)
Affinity DataKd:  1.10E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428239(CHEMBL2337448)
Affinity DataKd:  1.10E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428240(CHEMBL2337447)
Affinity DataKd:  1.80E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428241(CHEMBL2337446)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428242(CHEMBL2337445)
Affinity DataKd: >2.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428243(CHEMBL2337444)
Affinity DataKd: >2.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428244(CHEMBL2337443)
Affinity DataKd: >2.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428245(CHEMBL2337442)
Affinity DataKd: >2.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428235(CHEMBL2337028)
Affinity DataKd:  3.10E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428247(CHEMBL2337039)
Affinity DataKd:  1.58E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428248(CHEMBL2337038)
Affinity DataKd: >2.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428249(CHEMBL2337037)
Affinity DataKd: >2.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428250(CHEMBL2337036)
Affinity DataKd: >2.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428251(CHEMBL2337035)
Affinity DataKd:  7.00E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428252(CHEMBL2337034)
Affinity DataKd:  4.70E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428253(CHEMBL2337033)
Affinity DataKd: >2.00E+4nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428254(CHEMBL1609857)
Affinity DataKd:  6.90E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetWD repeat-containing protein 5(Human)
Entremed

Curated by ChEMBL
LigandPNGBDBM50428255(CHEMBL1231559)
Affinity DataIC50: 6.00E+3nMAssay Description:Antagonist activity at WDR5 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed