Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50005385
TargetTarget of rapamycin complex subunit LST8(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50491634(CHEMBL2386855)
Affinity DataIC50: 100nMAssay Description:Inhibition of mTORC1 in human PC3 cells assessed as reduction of phosphorylated 4E-BP1Thr37/46 level after 90 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetTarget of rapamycin complex subunit LST8(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50491633(CHEMBL2386856)
Affinity DataIC50: 100nMAssay Description:Inhibition of mTORC1 in human PC3 cells assessed as reduction of phosphorylated 4E-BP1Thr37/46 level after 90 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetTarget of rapamycin complex subunit LST8(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50491630(CHEMBL2386854)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of mTORC1 in human PC3 cells assessed as reduction of phosphorylated 4E-BP1Thr37/46 level after 90 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetTarget of rapamycin complex subunit LST8(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50491632(CHEMBL2386853)
Affinity DataIC50: 1.86E+3nMAssay Description:Inhibition of mTORC1 in human PC3 cells assessed as reduction of phosphorylated 4E-BP1Thr37/46 level after 90 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetTarget of rapamycin complex subunit LST8(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50491631(CHEMBL2386851)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mTORC1 in human PC3 cells assessed as reduction of phosphorylated 4E-BP1Thr37/46 level after 90 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetTarget of rapamycin complex subunit LST8(Human)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50491629(CHEMBL3037783)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mTORC1 in human PC3 cells assessed as reduction of phosphorylated 4E-BP1Thr37/46 level after 90 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed