Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50044618
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM25013(4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3S...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of AKT1 (unknown origin) after 1 hr by Z'-LYTE kinase assay in presence of 75 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50313650(8-(4-(1-aminocyclobutyl)phenyl)-9-phenyl-[1,2,4]tr...)
Affinity DataIC50: 10nMAssay Description:Inhibition of AKT1 (unknown origin) after 1 hr by Z'-LYTE kinase assay in presence of 75 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50022549(CHEMBL3299032)
Affinity DataIC50: 200nMAssay Description:Inhibition of AKT1 (unknown origin) after 30 mins by scintillation counting analysis in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50022551(CHEMBL3298512)
Affinity DataIC50: 580nMAssay Description:Inhibition of AKT1 (unknown origin) after 1 hr by Z'-LYTE kinase assay in presence of 75 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50022559(CHEMBL3298516)
Affinity DataIC50: 4.48E+3nMAssay Description:Inhibition of AKT1 (unknown origin) after 1 hr by Z'-LYTE kinase assay in presence of 75 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50022564(CHEMBL3298929)
Affinity DataIC50: 4.68E+3nMAssay Description:Inhibition of AKT1 (unknown origin) after 1 hr by Z'-LYTE kinase assay in presence of 75 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50022562(CHEMBL3298792)
Affinity DataIC50: 1.61E+4nMAssay Description:Inhibition of AKT1 (unknown origin) after 1 hr by Z'-LYTE kinase assay in presence of 75 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50022561(CHEMBL3298611)
Affinity DataIC50: 2.47E+4nMAssay Description:Inhibition of AKT1 (unknown origin) after 1 hr by Z'-LYTE kinase assay in presence of 75 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50022563(CHEMBL3298928)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of AKT1 (unknown origin) after 1 hr by Z'-LYTE kinase assay in presence of 75 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50022565(CHEMBL3298930)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of AKT1 (unknown origin) after 1 hr by Z'-LYTE kinase assay in presence of 75 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50022558(CHEMBL3298515)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of AKT1 (unknown origin) after 1 hr by Z'-LYTE kinase assay in presence of 75 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50022560(CHEMBL3298610)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of AKT1 (unknown origin) after 1 hr by Z'-LYTE kinase assay in presence of 75 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50022552(CHEMBL3298513)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of AKT1 (unknown origin) after 1 hr by Z'-LYTE kinase assay in presence of 75 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50022557(CHEMBL3298514)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of AKT1 (unknown origin) after 1 hr by Z'-LYTE kinase assay in presence of 75 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed