Compile Data Set for Download or QSAR
Report error Found 78 Enz. Inhib. hit(s) with all data for entry = 50045219
TargetMitogen-activated protein kinase 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050853(CHEMBL3318029)
Affinity DataIC50: 30nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetAurora kinase B(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050860(CHEMBL3318034)
Affinity DataIC50: 66nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetAurora kinase B(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050861(CHEMBL3318035)
Affinity DataIC50: 86nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetAurora kinase B(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050858(CHEMBL3318032)
Affinity DataIC50: 112nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetAurora kinase B(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050855(CHEMBL3318008)
Affinity DataIC50: 136nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetAurora kinase B(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050852(CHEMBL3318030)
Affinity DataIC50: 171nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050854(CHEMBL3318028)
Affinity DataIC50: 191nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetAurora kinase B(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050848(CHEMBL3318026)
Affinity DataIC50: 227nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetAurora kinase B(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050847(CHEMBL3318027)
Affinity DataIC50: 260nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050847(CHEMBL3318027)
Affinity DataIC50: 429nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetAurora kinase B(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050853(CHEMBL3318029)
Affinity DataIC50: 579nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetAurora kinase B(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050850(CHEMBL3318024)
Affinity DataIC50: 624nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050848(CHEMBL3318026)
Affinity DataIC50: 702nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetAurora kinase B(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050856(CHEMBL3318009)
Affinity DataIC50: 714nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050852(CHEMBL3318030)
Affinity DataIC50: 733nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050850(CHEMBL3318024)
Affinity DataIC50: 742nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetAurora kinase B(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050849(CHEMBL3318025)
Affinity DataIC50: 805nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050851(CHEMBL3318023)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetAurora kinase B(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050854(CHEMBL3318028)
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetAurora kinase B(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050859(CHEMBL3318033)
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetAurora kinase B(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050857(CHEMBL3318031)
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050849(CHEMBL3318025)
Affinity DataIC50: 1.72E+3nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetAurora kinase B(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050851(CHEMBL3318023)
Affinity DataIC50: 2.23E+3nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050847(CHEMBL3318027)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of TrkA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050847(CHEMBL3318027)
Affinity DataIC50: 6.05E+3nMAssay Description:Inhibition of c-Abl (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase Yes(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050847(CHEMBL3318027)
Affinity DataIC50: 7.95E+3nMAssay Description:Inhibition of YES (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050852(CHEMBL3318030)
Affinity DataIC50: 1.27E+4nMAssay Description:Inhibition of TrkA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050850(CHEMBL3318024)
Affinity DataIC50: 1.36E+4nMAssay Description:Inhibition of HIPK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050851(CHEMBL3318023)
Affinity DataIC50: 2.08E+4nMAssay Description:Inhibition of c-Abl (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase Yes(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050852(CHEMBL3318030)
Affinity DataIC50: 2.69E+4nMAssay Description:Inhibition of YES (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050853(CHEMBL3318029)
Affinity DataIC50: 3.16E+4nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050858(CHEMBL3318032)
Affinity DataIC50: 3.16E+4nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050854(CHEMBL3318028)
Affinity DataIC50: 3.16E+4nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050852(CHEMBL3318030)
Affinity DataIC50: 3.25E+4nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050851(CHEMBL3318023)
Affinity DataIC50: 3.71E+4nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase Yes(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050850(CHEMBL3318024)
Affinity DataIC50: 4.18E+4nMAssay Description:Inhibition of YES (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase Yes(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050848(CHEMBL3318026)
Affinity DataIC50: 4.29E+4nMAssay Description:Inhibition of YES (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050848(CHEMBL3318026)
Affinity DataIC50: 8.06E+4nMAssay Description:Inhibition of TrkA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase Yes(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050849(CHEMBL3318025)
Affinity DataIC50: 8.55E+4nMAssay Description:Inhibition of YES (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050848(CHEMBL3318026)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of c-Abl (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050851(CHEMBL3318023)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of TrkA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050852(CHEMBL3318030)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIPK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050854(CHEMBL3318028)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of TrkA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050853(CHEMBL3318029)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of TrkA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050847(CHEMBL3318027)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050850(CHEMBL3318024)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050850(CHEMBL3318024)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of c-Abl (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050849(CHEMBL3318025)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of c-Abl (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050849(CHEMBL3318025)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
TargetTyrosine-protein kinase Yes(Human)
University of Nantes

Curated by ChEMBL
LigandPNGBDBM50050853(CHEMBL3318029)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of YES (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
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