Compile Data Set for Download or QSAR
Report error Found 91 Enz. Inhib. hit(s) with all data for entry = 50044680
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025233(CHEMBL3330663)
Affinity DataEC50:  137nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50159165(2S,4aR,6a(R,7R,9S,10aS,10bR)-9-(acetyloxy)-2-(fura...)
Affinity DataEC50:  0.360nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025277(CHEMBL3330683)
Affinity DataEC50:  582nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025276(CHEMBL3330682)
Affinity DataEC50:  1.76E+3nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025275(CHEMBL3330681)
Affinity DataEC50:  1.21E+3nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025274(CHEMBL3330680)
Affinity DataEC50:  642nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025273(CHEMBL3330679)
Affinity DataEC50:  20nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025272(CHEMBL3330678)
Affinity DataEC50:  32nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025271(CHEMBL3330677)
Affinity DataEC50:  33nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025270(CHEMBL3330676)
Affinity DataEC50:  50nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025269(CHEMBL3330675)
Affinity DataEC50:  1.80E+3nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025268(CHEMBL3330674)
Affinity DataEC50:  27nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025266(CHEMBL3330672)
Affinity DataEC50:  21nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025265(CHEMBL3330671)
Affinity DataEC50:  10nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025264(CHEMBL3330670)
Affinity DataEC50:  7nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025261(CHEMBL3330669)
Affinity DataEC50:  37nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025260(CHEMBL3330668)
Affinity DataEC50:  477nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025255(CHEMBL3330667)
Affinity DataEC50:  23nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025237(CHEMBL3330666)
Affinity DataEC50:  11nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025235(CHEMBL3330665)
Affinity DataEC50:  25nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025234(CHEMBL3330664)
Affinity DataEC50:  698nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025267(CHEMBL3330673)
Affinity DataEC50:  38nMAssay Description:Inhibition of human kappa opioid receptor expressed in HEK293T cells assessed as inhibition of cAMP production after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50370067(CHEMBL1237164 | US12215173, Compound Naltrindole)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMu-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM21015([tyrosyl-3,5-3H(N)]-D-Ala2-Mephe4-glyol5-enkephali...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50159165(2S,4aR,6a(R,7R,9S,10aS,10bR)-9-(acetyloxy)-2-(fura...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025235(CHEMBL3330665)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025264(CHEMBL3330670)
Affinity DataKi:  9.60nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025255(CHEMBL3330667)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025277(CHEMBL3330683)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025233(CHEMBL3330663)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025237(CHEMBL3330666)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025261(CHEMBL3330669)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50170670((3S,4aR,4bS,6S,8R,8aR,10aR)-3-Furan-3-yl-4a,8a-dim...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025264(CHEMBL3330670)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025265(CHEMBL3330671)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025273(CHEMBL3330679)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025266(CHEMBL3330672)
Affinity DataKi:  135nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025271(CHEMBL3330677)
Affinity DataKi:  148nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025260(CHEMBL3330668)
Affinity DataKi:  153nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025268(CHEMBL3330674)
Affinity DataKi:  162nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025277(CHEMBL3330683)
Affinity DataKi:  228nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025272(CHEMBL3330678)
Affinity DataKi:  281nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025234(CHEMBL3330664)
Affinity DataKi:  284nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025277(CHEMBL3330683)
Affinity DataKi:  304nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025270(CHEMBL3330676)
Affinity DataKi:  323nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025276(CHEMBL3330682)
Affinity DataKi:  334nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025235(CHEMBL3330665)
Affinity DataKi:  362nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025234(CHEMBL3330664)
Affinity DataKi:  385nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025261(CHEMBL3330669)
Affinity DataKi:  439nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50025237(CHEMBL3330666)
Affinity DataKi:  540nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) expressed in HEK293T cells after 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2016
Entry Details Article
PubMed
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