Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50044716
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50027369(CHEMBL3342444)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human CD38 catalytic domain assessed as reduction in cADPR hydrolysis incubated for 10 mins by fluorimetric cycling assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50027370(CHEMBL3342440)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of human CD38 catalytic domain assessed as reduction in cADPR hydrolysis incubated for 10 mins by fluorimetric cycling assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50027374(CHEMBL3342443)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of human CD38 catalytic domain assessed as reduction in cADPR hydrolysis incubated for 10 mins by fluorimetric cycling assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50027373(CHEMBL3342442)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human CD38 catalytic domain assessed as reduction in cADPR hydrolysis incubated for 10 mins by fluorimetric cycling assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50027372(CHEMBL3342441)
Affinity DataIC50: 1.58E+5nMAssay Description:Inhibition of human CD38 catalytic domain assessed as reduction in cADPR hydrolysis incubated for 10 mins by fluorimetric cycling assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed
TargetADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1(Human)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50027371(Cyclic Inosine 5''-Diphosphoribose | CHEMBL1161863)
Affinity DataIC50: 2.76E+5nMAssay Description:Inhibition of human CD38 catalytic domain assessed as reduction in cADPR hydrolysis incubated for 10 mins by fluorimetric cycling assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2016
Entry Details Article
PubMed