Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50046285
TargetMonocarboxylate transporter 1(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50103571(CHEMBL3335793)
Affinity DataKd:  1.60nMAssay Description:Binding affinity to MCT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50103568(CHEMBL3335794)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50103567(CHEMBL3335792)
Affinity DataIC50: 5nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50425797(CHEMBL2316885)
Affinity DataIC50: 120nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMed
Target6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50445946(CHEMBL3105836)
Affinity DataIC50: 207nMAssay Description:Inhibition of PFKFB3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMed
TargetHexokinase-2(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50103565(CHEMBL3335788)
Affinity DataIC50: 316nMAssay Description:Inhibition of hexokinase 2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50433843(CHEMBL2382401)
Affinity DataIC50: 480nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50441138(CHEMBL2430727)
Affinity DataIC50: 500nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMed
TargetAlpha-enolase(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50103566(CHEMBL3335790)
Affinity DataIC50: 576nMAssay Description:Inhibition of ENO1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50052254(2',6'-dichloro-4-((2-chlorophenyl)thio)-5-...)
Affinity DataIC50: 870nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase B chain(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50052254(2',6'-dichloro-4-((2-chlorophenyl)thio)-5-...)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of LDHB (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMed
Target6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50445944(CHEMBL3105839)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of PFKFB3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50103570(CHEMBL3335796)
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of LDHA (unknown origin) by pyruvate competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMed
TargetPhosphoglycerate mutase 1(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50103572(CHEMBL3335789)
Affinity DataIC50: 1.31E+4nMAssay Description:Inhibition of PGM1 (unknown origin) by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50103570(CHEMBL3335796)
Affinity DataIC50: 1.47E+4nMAssay Description:Inhibition of LDHA (unknown origin) by NADH competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMed
Target6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50445948(CHEMBL3105848)
Affinity DataIC50: 2.29E+4nMAssay Description:Inhibition of PFKFB3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50103568(CHEMBL3335794)
Affinity DataKi:  4.80nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMed
TargetPhosphoglycerate mutase 1(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50103572(CHEMBL3335789)
Affinity DataKi:  3.91E+3nMAssay Description:Inhibition of PGM1 (unknown origin) by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50103570(CHEMBL3335796)
Affinity DataKi:  5.10E+3nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50103569(CHEMBL3335795)
Affinity DataKi:  3.78E+4nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2016
Entry Details Article
PubMed