Compile Data Set for Download or QSAR
Report error Found 93 Enz. Inhib. hit(s) with all data for entry = 50044818
TargetMelanocyte-stimulating hormone receptor(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataEC50:  0.0300nMAssay Description:Activity at mouse MC1R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031479(CHEMBL3358545)
Affinity DataEC50:  0.0420nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031473(CHEMBL3358549)
Affinity DataEC50:  0.0450nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031473(CHEMBL3358549)
Affinity DataEC50:  0.0480nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031479(CHEMBL3358545)
Affinity DataEC50:  0.0510nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031488(CHEMBL3358541)
Affinity DataEC50:  0.0510nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031488(CHEMBL3358541)
Affinity DataEC50:  0.0580nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataEC50:  0.0600nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031469(CHEMBL3358552)
Affinity DataEC50:  0.0670nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031469(CHEMBL3358552)
Affinity DataEC50:  0.0700nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031473(CHEMBL3358549)
Affinity DataEC50:  0.0740nMAssay Description:Activity at mouse MC1R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031492(CHEMBL3358539)
Affinity DataEC50:  0.0860nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031478(CHEMBL3358546)
Affinity DataEC50:  0.0870nMAssay Description:Activity at mouse MC1R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  0.0920nMAssay Description:Activity at mouse MC1R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031492(CHEMBL3358539)
Affinity DataEC50:  0.0980nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031479(CHEMBL3358545)
Affinity DataEC50:  0.100nMAssay Description:Activity at mouse MC1R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031486(CHEMBL3358544)
Affinity DataEC50:  0.110nMAssay Description:Activity at mouse MC1R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031496(CHEMBL3358535)
Affinity DataEC50:  0.130nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031496(CHEMBL3358535)
Affinity DataEC50:  0.130nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031490(CHEMBL3358540)
Affinity DataEC50:  0.130nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031478(CHEMBL3358546)
Affinity DataEC50:  0.130nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031478(CHEMBL3358546)
Affinity DataEC50:  0.140nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031471(CHEMBL3358550)
Affinity DataEC50:  0.140nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031470(CHEMBL3358551)
Affinity DataEC50:  0.140nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031490(CHEMBL3358540)
Affinity DataEC50:  0.140nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031470(CHEMBL3358551)
Affinity DataEC50:  0.150nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031471(CHEMBL3358550)
Affinity DataEC50:  0.150nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataEC50:  0.180nMAssay Description:Activity at mouse MC3R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031495(CHEMBL3358536)
Affinity DataEC50:  0.180nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataEC50:  0.190nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031495(CHEMBL3358536)
Affinity DataEC50:  0.190nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031478(CHEMBL3358546)
Affinity DataEC50:  0.200nMAssay Description:Activity at mouse MC3R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031469(CHEMBL3358552)
Affinity DataEC50:  0.200nMAssay Description:Activity at mouse MC1R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031473(CHEMBL3358549)
Affinity DataEC50:  0.200nMAssay Description:Activity at mouse MC3R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  0.200nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031479(CHEMBL3358545)
Affinity DataEC50:  0.210nMAssay Description:Activity at mouse MC3R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031500(CHEMBL2372859)
Affinity DataEC50:  0.210nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031486(CHEMBL3358544)
Affinity DataEC50:  0.220nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031489(CHEMBL3352878)
Affinity DataEC50:  0.230nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031494(CHEMBL3358537)
Affinity DataEC50:  0.240nMAssay Description:Activity at mouse MC1R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031488(CHEMBL3358541)
Affinity DataEC50:  0.25nMAssay Description:Activity at mouse MC1R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031486(CHEMBL3358544)
Affinity DataEC50:  0.290nMAssay Description:Activity at mouse MC3R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031469(CHEMBL3358552)
Affinity DataEC50:  0.290nMAssay Description:Activity at mouse MC3R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031489(CHEMBL3352878)
Affinity DataEC50:  0.290nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031499(CHEMBL3358542)
Affinity DataEC50:  0.310nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031470(CHEMBL3358551)
Affinity DataEC50:  0.320nMAssay Description:Activity at mouse MC1R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031486(CHEMBL3358544)
Affinity DataEC50:  0.340nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031492(CHEMBL3358539)
Affinity DataEC50:  0.360nMAssay Description:Activity at mouse MC1R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031488(CHEMBL3358541)
Affinity DataEC50:  0.440nMAssay Description:Activity at mouse MC3R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Mouse)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031498(CHEMBL3358533)
Affinity DataEC50:  0.460nMAssay Description:Activity at mouse MC1R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
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