Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50044875
TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034512(CHEMBL3359273)
Affinity DataEC50:  1.21E+4nMAssay Description:Positive allosteric modulation of human recombinant GLP1 receptor expressed in 9-3-H cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034510(CHEMBL3359272)
Affinity DataEC50:  3.00E+4nMAssay Description:Positive allosteric modulation of human recombinant GLP1 receptor expressed in 9-3-H cells by calcium mobilization assay in presence of EC20 of lirag...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034510(CHEMBL3359272)
Affinity DataEC50:  8.40E+3nMAssay Description:Positive allosteric modulation of human recombinant GLP1 receptor expressed in 9-3-H cells by calcium mobilization assay in presence of EC20 of exena...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034510(CHEMBL3359272)
Affinity DataEC50:  1.80E+3nMAssay Description:Positive allosteric modulation of human recombinant GLP1 receptor expressed in 9-3-H cells by calcium mobilization assay in presence of EC20 of GLP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034515(CHEMBL3359275)
Affinity DataEC50:  1.81E+4nMAssay Description:Positive allosteric modulation of human recombinant GLP1 receptor expressed in 9-3-H cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034514(CHEMBL3359274)
Affinity DataEC50:  1.03E+4nMAssay Description:Positive allosteric modulation of human recombinant GLP1 receptor expressed in 9-3-H cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034500(CHEMBL3359269)
Affinity DataEC50:  4.17E+3nMAssay Description:Positive allosteric modulation of human recombinant GLP1 receptor expressed in 9-3-H cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034510(CHEMBL3359272)
Affinity DataEC50:  1.30E+3nMAssay Description:Positive allosteric modulation of human recombinant GLP1 receptor expressed in 9-3-H cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034506(CHEMBL3359271)
Affinity DataEC50:  6.50E+3nMAssay Description:Positive allosteric modulation of human recombinant GLP1 receptor expressed in 9-3-H cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034505(CHEMBL3359270)
Affinity DataEC50:  2.04E+3nMAssay Description:Positive allosteric modulation of human recombinant GLP1 receptor expressed in 9-3-H cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034510(CHEMBL3359272)
Affinity DataEC50:  3.16E+4nMAssay Description:Positive allosteric modulation of human recombinant GLP1 receptor expressed in 9-3-H cells by calcium mobilization assay in presence of EC20 of lirag...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034505(CHEMBL3359270)
Affinity DataEC50:  2.04E+3nMAssay Description:Positive allosteric modulation of human recombinant GLP1 receptor expressed in 9-3-H cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034506(CHEMBL3359271)
Affinity DataEC50:  6.61E+3nMAssay Description:Positive allosteric modulation of human recombinant GLP1 receptor expressed in 9-3-H cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034510(CHEMBL3359272)
Affinity DataEC50:  1.32E+3nMAssay Description:Positive allosteric modulation of human recombinant GLP1 receptor expressed in 9-3-H cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034512(CHEMBL3359273)
Affinity DataEC50:  1.20E+4nMAssay Description:Positive allosteric modulation of human recombinant GLP1 receptor expressed in 9-3-H cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034514(CHEMBL3359274)
Affinity DataEC50:  1.02E+4nMAssay Description:Positive allosteric modulation of human recombinant GLP1 receptor expressed in 9-3-H cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034515(CHEMBL3359275)
Affinity DataEC50:  1.82E+4nMAssay Description:Positive allosteric modulation of human recombinant GLP1 receptor expressed in 9-3-H cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034510(CHEMBL3359272)
Affinity DataEC50:  1.82E+3nMAssay Description:Positive allosteric modulation of human recombinant GLP1 receptor expressed in 9-3-H cells by calcium mobilization assay in presence of EC20 of GLP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034510(CHEMBL3359272)
Affinity DataEC50:  8.51E+3nMAssay Description:Positive allosteric modulation of human recombinant GLP1 receptor expressed in 9-3-H cells by calcium mobilization assay in presence of EC20 of exena...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034500(CHEMBL3359269)
Affinity DataEC50:  4.10E+3nMAssay Description:Positive allosteric modulation of human recombinant GLP1 receptor expressed in 9-3-H cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034505(CHEMBL3359270)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034510(CHEMBL3359272)
Affinity DataIC50: 3.89E+3nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034510(CHEMBL3359272)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034505(CHEMBL3359270)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034505(CHEMBL3359270)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034505(CHEMBL3359270)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034510(CHEMBL3359272)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Vanderbilt University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50034510(CHEMBL3359272)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed