Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50044961
TargetAurora kinase B(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataKd:  3.10nMAssay Description:Binding affinity to AURKB (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataKd:  1.30nMAssay Description:Binding affinity to AURKA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataIC50: 735nMAssay Description:Inhibition of recombinant AURKB (unknown origin) after 60 mins by z'-lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataIC50: 1.34E+3nMAssay Description:Inhibition of recombinant AURKA (unknown origin) after 60 mins by z'-lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataIC50: 2.63E+3nMAssay Description:Inhibition of recombinant GSK-3 beta (unknown origin) after 60 mins by z'-lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of recombinant FLT1 (unknown origin) after 60 mins by z'-lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetPlatelet-derived growth factor receptor alpha(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataIC50: 4.04E+3nMAssay Description:Inhibition of recombinant PDGFR alpha (unknown origin) after 60 mins by z'-lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetAurora kinase C(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataIC50: 4.75E+3nMAssay Description:Inhibition of recombinant AURKC (unknown origin) after 60 mins by z'-lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 3(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataIC50: 5.19E+3nMAssay Description:Inhibition of recombinant FLT4 (unknown origin) after 60 mins by z'-lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataIC50: 5.96E+3nMAssay Description:Inhibition of recombinant KDR (unknown origin) after 60 mins by z'-lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek1(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of recombinant NEK1 (unknown origin) after 60 mins by z'-lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataIC50: 2.68E+4nMAssay Description:Inhibition of recombinant PKC alpha (unknown origin) after 60 mins by z'-lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataIC50: 3.86E+4nMAssay Description:Inhibition of recombinant AKT1 (unknown origin) after 60 mins by z'-lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetCasein kinase I isoform alpha(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataIC50: 7.88E+4nMAssay Description:Inhibition of recombinant CK1 alpha1 (unknown origin) after 60 mins by z'-lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant PRKACA (unknown origin) after 60 mins by z'-lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant EGFR (unknown origin) after 60 mins by z'-lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetInsulin-like growth factor 1 receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant IGF1R (unknown origin) after 60 mins by z'-lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant MAPK1 (unknown origin) after 60 mins by z'-lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 2(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant PAK2 (unknown origin) after 60 mins by z'-lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50038423(CHEMBL3361128)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant PLK1 (unknown origin) after 60 mins by z'-lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed