Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50044974
TargetBifunctional ligase/repressor BirA(Escherichia coli (strain K12))
University of Nebraska-Lincoln

Curated by ChEMBL
LigandPNGBDBM50039492(CHEMBL1231498)
Affinity DataKd:  1.5nMAssay Description:Binding affinity to Escherichia coli biotin protein ligaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetBiotin--protein ligase(Human)
University of Nebraska-Lincoln

Curated by ChEMBL
LigandPNGBDBM50039492(CHEMBL1231498)
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of human recombinant HLCS using P67 as substrate after 2 hrs relative to vehicle-treated controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetBiotin--protein ligase(Human)
University of Nebraska-Lincoln

Curated by ChEMBL
LigandPNGBDBM50039493(CHEMBL3357333)
Affinity DataIC50: 3.97E+4nMAssay Description:Inhibition of human recombinant HLCS using P67 as substrate after 2 hrs relative to vehicle-treated controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetBiotin--protein ligase(Human)
University of Nebraska-Lincoln

Curated by ChEMBL
LigandPNGBDBM50039494(CHEMBL3357334)
Affinity DataIC50: 2.04E+5nMAssay Description:Inhibition of human recombinant HLCS using P67 as substrate after 2 hrs relative to vehicle-treated controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetBiotin--protein ligase(Human)
University of Nebraska-Lincoln

Curated by ChEMBL
LigandPNGBDBM50039493(CHEMBL3357333)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of human recombinant HLCS using P67 as substrate after 2 hrs relative to vehicle-treated controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetBiotin--protein ligase(Human)
University of Nebraska-Lincoln

Curated by ChEMBL
LigandPNGBDBM50039494(CHEMBL3357334)
Affinity DataKi:  1.04E+4nMAssay Description:Inhibition of human recombinant HLCS using P67 as substrate after 2 hrs relative to vehicle-treated controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed
TargetBiotin--protein ligase(Human)
University of Nebraska-Lincoln

Curated by ChEMBL
LigandPNGBDBM50039492(CHEMBL1231498)
Affinity DataKi:  7.54E+5nMAssay Description:Inhibition of human recombinant HLCS using P67 as substrate after 2 hrs relative to vehicle-treated controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/17/2016
Entry Details Article
PubMed