Compile Data Set for Download or QSAR
Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 50006240
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498068(CHEMBL3394234)
Affinity DataIC50: 1nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498093(CHEMBL3394236)
Affinity DataIC50: 2nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498069(CHEMBL3394233)
Affinity DataIC50: 2nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498070(CHEMBL3394163)
Affinity DataIC50: 3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498096(CHEMBL3394232)
Affinity DataIC50: 5nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498082(CHEMBL3394237)
Affinity DataIC50: 5nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498089(CHEMBL3394162)
Affinity DataIC50: 6nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498090(CHEMBL3394161)
Affinity DataIC50: 6nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498057(CHEMBL3394235)
Affinity DataIC50: 17nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498060(CHEMBL3394249)
Affinity DataIC50: 22nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498059(CHEMBL3394250)
Affinity DataIC50: 32nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498061(CHEMBL3394247)
Affinity DataIC50: 100nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498062(CHEMBL3394246)
Affinity DataIC50: 140nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498056(CHEMBL3394242)
Affinity DataIC50: 200nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498080(CHEMBL3394245)
Affinity DataIC50: 240nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498074(CHEMBL3394155)
Affinity DataIC50: 250nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498079(CHEMBL3394248)
Affinity DataIC50: 330nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498088(CHEMBL3394240)
Affinity DataIC50: 350nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498085(CHEMBL3394151)
Affinity DataIC50: 420nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498073(CHEMBL3394157)
Affinity DataIC50: 430nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498063(CHEMBL3394244)
Affinity DataIC50: 820nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498065(CHEMBL3394241)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498058(CHEMBL3394153)
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498094(CHEMBL3394154)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498091(CHEMBL3394160)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498077(CHEMBL3394148)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498078(CHEMBL3394146)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498054(CHEMBL1477426)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498064(CHEMBL3394243)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498084(CHEMBL3394156)
Affinity DataIC50: 2.63E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498095(CHEMBL3394152)
Affinity DataIC50: 2.73E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498055(CHEMBL3394145)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498076(CHEMBL3394149)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498072(CHEMBL3394158)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498083(CHEMBL3394159)
Affinity DataIC50: 1.43E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498075(CHEMBL3394150)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498087(CHEMBL3394251)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498092(CHEMBL3394252)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498071(CHEMBL110569)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498086(CHEMBL3394147)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498081(CHEMBL3394239)
Affinity DataIC50: 1.33E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498067(CHEMBL3394238)
Affinity DataIC50: 5.90E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetThymidylate kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50498066(CHEMBL356501)
Affinity DataIC50: 6.34E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed