Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50045029
TargetAcetylcholinesterase(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50042282(CHEMBL3361270)
Affinity DataIC50: 160nMAssay Description:Inhibition of AChE (unknown origin) assessed as reduction in acetylthiocholine iodide hydrolysis after 15 mins by Ellman methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50042284(CHEMBL3361277)
Affinity DataIC50: 930nMAssay Description:Inhibition of BuChE (unknown origin) assessed as reduction in S-butyrylthiocholine chloride hydrolysis after 15 mins by Ellman methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50042282(CHEMBL3361270)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of BuChE (unknown origin) assessed as reduction in S-butyrylthiocholine chloride hydrolysis after 15 mins by Ellman methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM10404(galantamine | (1S,12S,14R)-9-methoxy-4-methyl-11-o...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of AChE (unknown origin) assessed as reduction in acetylthiocholine iodide hydrolysis after 15 mins by Ellman methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM29278(Saccharimide | SAC | Garantose | CHEMBL310671 | Sa...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of BuChE (unknown origin) assessed as reduction in S-butyrylthiocholine chloride hydrolysis after 15 mins by Ellman methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetCholinesterase(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50042283(CHEMBL3361265)
Affinity DataIC50: 5.08E+3nMAssay Description:Inhibition of BuChE (unknown origin) assessed as reduction in S-butyrylthiocholine chloride hydrolysis after 15 mins by Ellman methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed