Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50045615
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
The University of Georgia
Curated by ChEMBL
The University of Georgia
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
The University of Georgia
Curated by ChEMBL
The University of Georgia
Curated by ChEMBL
Affinity DataIC50: 610nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
The University of Georgia
Curated by ChEMBL
The University of Georgia
Curated by ChEMBL
Affinity DataIC50: 1.15E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
The University of Georgia
Curated by ChEMBL
The University of Georgia
Curated by ChEMBL
Affinity DataIC50: 1.25E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT5 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
Affinity DataIC50: 1.74E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT8 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
The University of Georgia
Curated by ChEMBL
The University of Georgia
Curated by ChEMBL
Affinity DataIC50: 1.81E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
The University of Georgia
Curated by ChEMBL
The University of Georgia
Curated by ChEMBL
Affinity DataIC50: 2.03E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
The University of Georgia
Curated by ChEMBL
The University of Georgia
Curated by ChEMBL
Affinity DataIC50: 2.37E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
The University of Georgia
Curated by ChEMBL
The University of Georgia
Curated by ChEMBL
Affinity DataIC50: 2.56E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
The University of Georgia
Curated by ChEMBL
The University of Georgia
Curated by ChEMBL
Affinity DataIC50: 2.67E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
The University of Georgia
Curated by ChEMBL
The University of Georgia
Curated by ChEMBL
Affinity DataIC50: 3.05E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
The University of Georgia
Curated by ChEMBL
The University of Georgia
Curated by ChEMBL
Affinity DataIC50: 3.38E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
The University of Georgia
Curated by ChEMBL
The University of Georgia
Curated by ChEMBL
Affinity DataIC50: 3.39E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
The University of Georgia
Curated by ChEMBL
The University of Georgia
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
The University of Georgia
Curated by ChEMBL
The University of Georgia
Curated by ChEMBL
Affinity DataIC50: 5.76E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
Affinity DataIC50: 5.80E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged CARM1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
The University of Georgia
Curated by ChEMBL
The University of Georgia
Curated by ChEMBL
Affinity DataIC50: 6.43E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
Affinity DataIC50: 7.04E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT5 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
Affinity DataIC50: 7.23E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged CARM1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
Affinity DataIC50: 8.36E+3nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT5 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
Affinity DataIC50: 2.15E+4nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged CARM1 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
Affinity DataIC50: 2.84E+4nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT8 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
Affinity DataIC50: 3.54E+4nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT5 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
Affinity DataIC50: 8.49E+4nMAssay Description:Displacement of [3H]-SAM from recombinant His6-tagged PRMT8 (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 5 mins prior to H4...More data for this Ligand-Target Pair
