Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50006247
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498143(CHEMBL3407602)
Affinity DataIC50: 31nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498128(CHEMBL3410944)
Affinity DataIC50: 35nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498142(CHEMBL3407601)
Affinity DataIC50: 38nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498137(CHEMBL3410941)
Affinity DataIC50: 47nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498150(CHEMBL3407599)
Affinity DataIC50: 79nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498135(CHEMBL3407603)
Affinity DataIC50: 94nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498134(CHEMBL3407605)
Affinity DataIC50: 96nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498147(CHEMBL3407604)
Affinity DataIC50: 101nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498141(CHEMBL3407597)
Affinity DataIC50: 118nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498130(CHEMBL3407600)
Affinity DataIC50: 121nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498140(CHEMBL3407596)
Affinity DataIC50: 123nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498144(CHEMBL3407608)
Affinity DataIC50: 158nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498133(CHEMBL3407606)
Affinity DataIC50: 173nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498151(CHEMBL3407598)
Affinity DataIC50: 178nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498132(CHEMBL3407612)
Affinity DataIC50: 187nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498131(CHEMBL3407613)
Affinity DataIC50: 230nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498149(CHEMBL3407594)
Affinity DataIC50: 248nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498127(CHEMBL3407607)
Affinity DataIC50: 251nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498145(CHEMBL3407593)
Affinity DataIC50: 258nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498152(CHEMBL3407611)
Affinity DataIC50: 263nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498129(CHEMBL3407609)
Affinity DataIC50: 279nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498139(CHEMBL3407592)
Affinity DataIC50: 350nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498138(CHEMBL3410945)
Affinity DataIC50: 352nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498136(CHEMBL3410942)
Affinity DataIC50: 554nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498146(CHEMBL3407610)
Affinity DataIC50: 642nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498153(CHEMBL3407595)
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498154(CHEMBL3407614)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50498148(CHEMBL3410943)
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibition of human recombinant KDM1A/CoREST complex expressed in Escherichia coli using mono-methylated H3-K4 peptide containing 21 amino acids as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed