Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50045440
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50062743(CHEMBL3397787)
Affinity DataIC50: 25nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-inducted alkaline phosphatase expression after 24 hrs by plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50062741(CHEMBL3397781)
Affinity DataIC50: 26nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-inducted alkaline phosphatase expression after 24 hrs by plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50062751(CHEMBL3397788)
Affinity DataIC50: 36nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-inducted alkaline phosphatase expression after 24 hrs by plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50062747(CHEMBL3397782)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-inducted alkaline phosphatase expression after 24 hrs by plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50062741(CHEMBL3397781)
Affinity DataIC50: 53nMAssay Description:Displacement of [1,2,6,7-3H]progesterone from human recombinant PR LBD after 24 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50062745(CHEMBL3397778)
Affinity DataIC50: 53nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-inducted alkaline phosphatase expression after 24 hrs by plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50062746(CHEMBL3397780)
Affinity DataIC50: 58nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-inducted alkaline phosphatase expression after 24 hrs by plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50062739(CHEMBL3397790)
Affinity DataIC50: 74nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-inducted alkaline phosphatase expression after 24 hrs by plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50062738(CHEMBL3397789)
Affinity DataIC50: 119nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-inducted alkaline phosphatase expression after 24 hrs by plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50062749(CHEMBL3397784)
Affinity DataIC50: 125nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-inducted alkaline phosphatase expression after 24 hrs by plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50062748(CHEMBL3397783)
Affinity DataIC50: 174nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-inducted alkaline phosphatase expression after 24 hrs by plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50062744(CHEMBL3397779)
Affinity DataIC50: 178nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-inducted alkaline phosphatase expression after 24 hrs by plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50062742(CHEMBL3397786)
Affinity DataIC50: 228nMAssay Description:Displacement of [1,2,6,7-3H]progesterone from human recombinant PR LBD after 24 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50062742(CHEMBL3397786)
Affinity DataIC50: 311nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-inducted alkaline phosphatase expression after 24 hrs by plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50062750(CHEMBL3397785)
Affinity DataIC50: 404nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-inducted alkaline phosphatase expression after 24 hrs by plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50062740(CHEMBL3397791)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at PR in human T47D cells assessed as inhibition of progesterone-inducted alkaline phosphatase expression after 24 hrs by plate r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50062743(CHEMBL3397787)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [1,2,6,7-3H]progesterone from human recombinant PR LBD after 24 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed